日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Protein tyrosine phosphatase inactivation by electrophilic tyrosine modification

亲电酪氨酸修饰导致蛋白质酪氨酸磷酸酶失活

Ware, Madeleine L; Leace, David M; Qu, Zihan; Schaefer, Quentin; Vaidya, Sagar D; Horvath, Mikayla L; Li, Zhihong; Bai, Yunpeng; Zhang, Zhong-Yin; Hsu, Ku-Lung

In Cellulo pharmacological profiling and genomic editing reveals paralog-specific targets for PA generation during PLC signaling.

在 Cellulo 中,药理学分析和基因组编辑揭示了 PLC 信号传导过程中 PA 生成的旁系同源特异性靶点。

Weckerly Claire C, Murtagh Olivia L, Swayhoover Tiernan, Pemberton Joshua G, Hsu Ku-Lung, Hammond Gerald R V

Advancing Covalent Ligand and Drug Discovery beyond Cysteine

推进半胱氨酸以外的共价配体和药物发现

Kim, Gibae; Grams, R Justin; Hsu, Ku-Lung

A Glutathione S-Transferase Pi Molecular Glue Tethers Splicing Factors and Remodels Cell Metabolism

谷胱甘肽S-转移酶Pi分子胶连接剪接因子并重塑细胞代谢

Leace, David M; Ware, Madeleine L; Murtagh, Olivia; Tsai, Hsiao-Kuei; Chang, Chin-Yuan; Hsu, Ku-Lung

Acetaminophen inhibits diacylglycerol lipase synthesis of 2-arachidonoyl glycerol: Implications for nociception

对乙酰氨基酚抑制二酰甘油脂肪酶合成2-花生四烯酸甘油酯:对伤害感受的影响

Dvorakova, Michaela; Bosquez-Berger, Taryn; Billingsley, Jenna; Murataeva, Natalia; Woodward, Taylor; Leishman, Emma; Zimmowitch, Anaëlle; Gibson, Anne; Wager-Miller, Jim; Cai, Ruyi; Cai, Shangxuan; Ware, Tim; Hsu, Ku-Lung; Li, Yulong; Bradshaw, Heather; Mackie, Ken; Straiker, Alex

Discovery and Optimization of a Covalent AKR1C3 Inhibitor

共价AKR1C3抑制剂的发现与优化

Grams, R Justin; Wolfe, Wesley J; Seal, Robert J; Veccia, James; Hsu, Ku-Lung

Emerging opportunities for intact and native protein analysis using chemical proteomics

利用化学蛋白质组学进行完整天然蛋白质分析的新机遇

Edwards, Alexis N; Hsu, Ku-Lung

Characterization of Mast2 kinase defines structural features, regulation, and substrates

Mast2激酶的特性分析阐明了其结构特征、调控机制和底物。

Lemke, Michael C; Chen, Miaomiao; Jang, Sophia S; Rader, Michael T; Avala, Nithin R; Bauchle, Casey J; Pluguez, Rafael; Miller, Ciara J; Butler, John D; Hargett, Stefan R; Lank, Daniel S; Seltzer, Brandon D; Stornetta, Daniel S; Fu, Zheng; Hsu, Ku-Lung; Harris, Thurl E

Human PTGR2 Inactivation Alters Eicosanoid Metabolism and Cytokine Response of Inflammatory Macrophages

人类PTGR2失活会改变炎症巨噬细胞的类花生酸代谢和细胞因子反应

Founds, Michael W; Murtagh, Olivia L; Grams, R Justin; Li, Zhihong; Ciancone, Anthony M; Seal, Robert J; Hsu, Ku-Lung

Stereoselective Degradation of Diacylglycerol Kinases Potentiate T cell Activation and Tumor Cell Cytotoxicity

二酰甘油激酶的立体选择性降解可增强T细胞活化和肿瘤细胞毒性

Shaikh, Minhaj; Mookherjee, Surya Pravo; Weckerly, Claire C; Libby, Adam H; Xiao, Aizhen; Zhao, Yunge; Vaidya, Sagar D; Kim, AeRyon; Li, Zhihong; Ware, Madeleine L; Marants, Michelle; Murtagh, Olivia L; Wolfe, Wesley J; Bullock, Timothy Nj; Purow, Benjamin W; Hammond, Gerald R V; Hsu, Ku-Lung