日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification and characterization of a novel inhibitor of influenza A virus that acts by blocking nucleoprotein oligomerization

鉴定并表征了一种新型甲型流感病毒抑制剂,该抑制剂通过阻断核蛋白寡聚化发挥作用。

Leonard, Vincent H J; Vidales, Dianna B; Taft, Benjamin R; Hesse, Matthew J; Lee, Patrick S; Mamo, Mulugeta; Bussiere, Dirksen E; Wolff, Karen C; Kuhen, Kelli L; Wedel, Laura; Growcott, Ellena; Osborne, Colin; Octaviani, Cassio P; Huang, Pinghan; Tseng, Chien-Te Kent; Abend, Johanna R; Wong, Kelly A; Zhong, Weidong; Tully, David C; Ganem, Don

The ReFRAME library as a comprehensive drug repurposing library and its application to the treatment of cryptosporidiosis

ReFRAME 库作为一个综合性药物重定位库及其在隐孢子虫病治疗中的应用

Janes, Jeff; Young, Megan E; Chen, Emily; Rogers, Nicole H; Burgstaller-Muehlbacher, Sebastian; Hughes, Laura D; Love, Melissa S; Hull, Mitchell V; Kuhen, Kelli L; Woods, Ashley K; Joseph, Sean B; Petrassi, H Michael; McNamara, Case W; Tremblay, Matthew S; Su, Andrew I; Schultz, Peter G; Chatterjee, Arnab K

High-Throughput Assay and Discovery of Small Molecules that Interrupt Malaria Transmission

利用高通量检测方法发现能够阻断疟疾传播的小分子

Plouffe, David M; Wree, Melanie; Du, Alan Y; Meister, Stephan; Li, Fengwu; Patra, Kailash; Lubar, Aristea; Okitsu, Shinji L; Flannery, Erika L; Kato, Nobutaka; Tanaseichuk, Olga; Comer, Eamon; Zhou, Bin; Kuhen, Kelli; Zhou, Yingyao; Leroy, Didier; Schreiber, Stuart L; Scherer, Christina A; Vinetz, Joseph; Winzeler, Elizabeth A

Direct inhibitors of InhA are active against Mycobacterium tuberculosis

InhA 的直接抑制剂对结核分枝杆菌有效

Manjunatha, Ujjini H; S Rao, Srinivasa P; Kondreddi, Ravinder Reddy; Noble, Christian G; Camacho, Luis R; Tan, Bee H; Ng, Seow H; Ng, Pearly Shuyi; Ma, Ng L; Lakshminarayana, Suresh B; Herve, Maxime; Barnes, Susan W; Yu, Weixuan; Kuhen, Kelli; Blasco, Francesca; Beer, David; Walker, John R; Tonge, Peter J; Glynne, Richard; Smith, Paul W; Diagana, Thierry T

No robust evidence of lumefantrine resistance

尚无确凿证据表明存在卢美芬汀耐药性

Hamed, Kamal; Kuhen, Kelli

Mutations in the P-type cation-transporter ATPase 4, PfATP4, mediate resistance to both aminopyrazole and spiroindolone antimalarials

P型阳离子转运蛋白ATPase 4 (PfATP4) 的突变介导了对氨基吡唑和螺吲哚酮类抗疟药的耐药性。

Flannery, Erika L; McNamara, Case W; Kim, Sang Wan; Kato, Tomoyo Sakata; Li, Fengwu; Teng, Christine H; Gagaring, Kerstin; Manary, Micah J; Barboa, Rachel; Meister, Stephan; Kuhen, Kelli; Vinetz, Joseph M; Chatterjee, Arnab K; Winzeler, Elizabeth A

KAI407, a potent non-8-aminoquinoline compound that kills Plasmodium cynomolgi early dormant liver stage parasites in vitro

KAI407 是一种强效的非 8-氨基喹啉类化合物,可在体外杀死猴疟原虫早期休眠肝期寄生虫。

Zeeman, Anne-Marie; van Amsterdam, Sandra M; McNamara, Case W; Voorberg-van der Wel, Annemarie; Klooster, Els J; van den Berg, Alexander; Remarque, Edmond J; Plouffe, David M; van Gemert, Geert-Jan; Luty, Adrian; Sauerwein, Robert; Gagaring, Kerstin; Borboa, Rachel; Chen, Zhong; Kuhen, Kelli; Glynne, Richard J; Chatterjee, Arnab K; Nagle, Advait; Roland, Jason; Winzeler, Elizabeth A; Leroy, Didier; Campo, Brice; Diagana, Thierry T; Yeung, Bryan K S; Thomas, Alan W; Kocken, Clemens H M

KAF156 is an antimalarial clinical candidate with potential for use in prophylaxis, treatment, and prevention of disease transmission

KAF156 是一种抗疟临床候选药物,具有用于预防、治疗和防止疾病传播的潜力。

Kelli L Kuhen, Arnab K Chatterjee, Matthias Rottmann, Kerstin Gagaring, Rachel Borboa, Jennifer Buenviaje, Zhong Chen, Carolyn Francek, Tao Wu, Advait Nagle, S Whitney Barnes, David Plouffe, Marcus C S Lee, David A Fidock, Wouter Graumans, Marga van de Vegte-Bolmer, Geert J van Gemert, Grennady Wirj

Targeting Plasmodium PI(4)K to eliminate malaria

针对疟原虫PI(4)K消除疟疾

Case W McNamara #, Marcus Cs Lee #, Chek Shik Lim, Siau Hoi Lim, Jason Roland, Oliver Simon, Bryan Ks Yeung, Arnab K Chatterjee, Susan L McCormack, Micah J Manary, Anne-Marie Zeeman, Koen J Dechering, Tr Santha Kumar, Philipp P Henrich, Kerstin Gagaring, Maureen Ibanez, Nobutaka Kato, Kelli L Kuhen,

Imidazolopiperazines: lead optimization of the second-generation antimalarial agents

咪唑并哌嗪类:第二代抗疟药物的先导优化

Advait Nagle, Tao Wu, Kelli Kuhen, Kerstin Gagaring, Rachel Borboa, Caroline Francek, Zhong Chen, David Plouffe, Xuena Lin, Christopher Caldwell, Jared Ek, Suzanne Skolnik, Fenghua Liu, Jianling Wang, Jonathan Chang, Chun Li, Bo Liu, Thomas Hollenbeck, Tove Tuntland, John Isbell, Tiffany Chuan, Phil