日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design, synthesis, antitumor activities and biological studies of novel diaryl substituted fused heterocycles as dual ligands targeting tubulin and katanin

新型二芳基取代稠杂环化合物作为针对微管蛋白和剑蛋白的双配体的设计、合成、抗肿瘤活性及生物学研究

Feng Gao, Yuru Liang, Pengfei Zhou, Jiayi Cheng, Kuiling Ding, Yang Wang

Design, synthesis, biological evaluation and cocrystal structures with tubulin of chiral β-lactam bridged combretastatin A-4 analogues as potent antitumor agents

手性β-内酰胺桥联康普立停A-4类似物的设计、合成、生物学评价及与微管蛋白的共晶结构作为强效抗肿瘤药物

Pengfei Zhou, Yuru Liang, Hao Zhang, Hao Jiang, Kechang Feng, Pan Xu, Jie Wang, Xiaoming Wang, Kuiling Ding, Cheng Luo, Mingming Liu, Yang Wang