日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Dynamic signature of activity-stability tradeoff in lactamase evolution

内酰胺酶进化中活性-稳定性权衡的动态特征

Arcia, Ernesto; Keramisanou, Dimitra; Jacobs, Lian M C; Parker, McKenna; Delgado, Julián M; Kumar Mv, Vasantha; Varma, Sameer; Abzalimov, Rinat; Chen, Yu; Gelis, Ioannis

Chemical modulation of cytosolic BAX homodimer potentiates BAX activation and apoptosis

细胞浆 BAX 同型二聚体的化学调节增强 BAX 活化和细胞凋亡

Nadege Gitego, Bogos Agianian, Oi Wei Mak, Vasantha Kumar Mv, Emily H Cheng, Evripidis Gavathiotis

BCA101 Is a Tumor-Targeted Bifunctional Fusion Antibody That Simultaneously Inhibits EGFR and TGFβ Signaling to Durably Suppress Tumor Growth

BCA101 是一种针对肿瘤的双功能融合抗体,可同时抑制 EGFR 和 TGFβ 信号传导,从而持久抑制肿瘤生长

Srinivas Reddy Boreddy, Reshmi Nair, Prashant Kumar Pandey, Anshu Kuriakose, Shivakumar Bhadravathi Marigowda, Chaitali Dey, Arindam Banerjee, Hanumant Kulkarni, Milind Sagar, Shiv Ram Krishn, Shruthi Rao, Madhukara Ar, Vinita Tiwari, Bhavna Alke, Prashantha Kumar Mv, Meena Shri, Chaitrali Dhamne, S

Modulating mitofusins to control mitochondrial function and signaling

调节线粒体融合蛋白来控制线粒体功能和信号传导

Emmanouil Zacharioudakis, Bogos Agianian, Vasantha Kumar Mv, Nikolaos Biris, Thomas P Garner, Inna Rabinovich-Nikitin, Amanda T Ouchida, Victoria Margulets, Lars Ulrik Nordstrøm, Joel S Riley, Igor Dolgalev, Yun Chen, Andre J H Wittig, Ryan Pekson, Chris Mathew, Peter Wei, Aristotelis Tsirigos, Step

Molecular insights into the interaction of Hsp90 with allosteric inhibitors targeting the C-terminal domain

从分子层面深入了解 Hsp90 与靶向 C 端结构域的变构抑制剂的相互作用

Kumar Mv, Vasantha; Ebna Noor, Radwan; Davis, Rachel E; Zhang, Zheng; Sipavicius, Edvinas; Keramisanou, Dimitra; Blagg, Brian S J; Gelis, Ioannis