日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identifying interactions between TDP-43's N-terminal and RNA-binding domains

鉴定TDP-43 N端结构域与RNA结合结构域之间的相互作用

Scott, David D; Jena, Lipsa; Rajaram, Akash; Ang, Jason; Perez-Miller, Samantha; Kumirov, Vlad; Khanna, Rajesh; Khanna, May

Trifluoromethylation of Arenes and Heterocycles via a Bench-Stable Photocaged Trifluoromethylation Reagent

利用台式稳定的光笼三氟甲基化试剂对芳烃和杂环化合物进行三氟甲基化

Rustin, Gavin J; Agarwal, Vishal; Dalton, Penelope I; Jiang, Zenghui; Liu, Zhao; Najor, Isabella G; Heydari, Bahar; Heydari, Beeta; Kuehl, Nicholas J; Kumirov, Vlad; Taylor, Michael T; Gustafson, Jeffrey L

Structure-Based Design of Glycosylated Oxytocin Analogues with Improved Selectivity and Antinociceptive Activity

基于结构的糖基化催产素类似物设计及其选择性和镇痛活性的提高

Szabó, Lajos Z; Tanguturi, Parthasaradhireddy; Goodman, Hannah J; Sprőber, Sára; Liu, Chenxi; Al-Obeidi, Fahad; Bartlett, Mitchell J; Falk, Torsten; Kumirov, Vlad K; Heien, M Leandro; Streicher, John M; Polt, Robin

Peptide exchange on MHC-I by TAPBPR is driven by a negative allostery release cycle

TAPBPR 在 MHC-I 上进行的肽交换是由负变构释放循环驱动的

Andrew C McShan, Kannan Natarajan, Vlad K Kumirov, David Flores-Solis, Jiansheng Jiang, Mareike Badstübner, Jugmohit S Toor, Clive R Bagshaw, Evgenii L Kovrigin, David H Margulies, Nikolaos G Sgourakis

Multistep mutational transformation of a protein fold through structural intermediates

蛋白质折叠通过结构中间体发生多步突变转变

Kumirov, Vlad K; Dykstra, Emily M; Hall, Branwen M; Anderson, William J; Szyszka, Taylor N; Cordes, Matthew H J

An allosteric site in the T-cell receptor Cβ domain plays a critical signalling role

T细胞受体Cβ结构域中的变构位点发挥着关键的信号传导作用

Kannan Natarajan ,Andrew C McShan ,Jiansheng Jiang ,Vlad K Kumirov ,Rui Wang ,Huaying Zhao ,Peter Schuck ,Mulualem E Tilahun ,Lisa F Boyd ,Jinfa Ying ,Ad Bax ,David H Margulies ,Nikolaos G Sgourakis

Foldability of a Natural De Novo Evolved Protein

天然从头进化蛋白质的折叠性

Bungard, Dixie; Copple, Jacob S; Yan, Jing; Chhun, Jimmy J; Kumirov, Vlad K; Foy, Scott G; Masel, Joanna; Wysocki, Vicki H; Cordes, Matthew H J

Synthesis and Investigation of Mixed μ-Opioid and δ-Opioid Agonists as Possible Bivalent Ligands for Treatment of Pain

合成和研究混合型μ-阿片受体和δ-阿片受体激动剂作为治疗疼痛的潜在二价配体

Vardanyan, Ruben S; Cain, James P; Haghighi, Saghar Mowlazadeh; Kumirov, Vlad K; McIntosh, Mary I; Sandweiss, Alexander J; Porreca, Frank; Hruby, Victor J

Studying protein fold evolution with hybrids of differently folded homologs

利用不同折叠方式的同源蛋白杂交体研究蛋白质折叠进化

Eaton, Karen V; Anderson, William J; Dubrava, Matthew S; Kumirov, Vlad K; Dykstra, Emily M; Cordes, Matthew H J

Novel fentanyl-based dual μ/δ-opioid agonists for the treatment of acute and chronic pain

新型芬太尼类双重 μ/δ-阿片类激动剂用于治疗急性和慢性疼痛

Alexander T Podolsky, Alexander Sandweiss, Jackie Hu, Edward J Bilsky, Jim P Cain, Vlad K Kumirov, Yeon Sun Lee, Victor J Hruby, Ruben S Vardanyan, Todd W Vanderah