日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

New Insights of Muraymycin A1 and Its Analogs as DPAGT1 Inhibitors

Muraymycin A1及其类似物作为DPAGT1抑制剂的新见解

Mitachi, Katsuhiko; Daria, Deidre; Kirsh, Jacob M; Effah, Wendy; Narayanan, Ramesh; Clemons, William M Jr; Kurosu, Michio

DPAGT1-Perspective as an Anticancer Drug Target

DPAGT1——作为抗癌药物靶点的展望

Kurosu, Michio; Mitachi, Katsuhiko

Structures of bacterial and human phosphoglycosyltransferases bound to a common inhibitor inform selective therapeutics

细菌和人类磷酸糖基转移酶与共同抑制剂结合的结构为选择性治疗提供了信息

Kaudeer, Beebee Yusrah; Kirsh, Jacob M; Mitachi, Katsuhiko; Ochoa, Jessica M; Soroush-Pejrimovsky, Marie-Therese; Li, Yancheng E; Nguyen, Vy N; Kurosu, Michio; Clemons, William M Jr

An improved total synthesis of tunicamycin V

改进的衣霉素V全合成

Mitachi, Katsuhiko; Mingle, David; Kurosu, Michio

Concise Synthesis of Tunicamycin V and Discovery of a Cytostatic DPAGT1 Inhibitor

简洁合成衣霉素V及发现一种细胞抑制性DPAGT1抑制剂

Mitachi, Katsuhiko; Mingle, David; Effah, Wendy; Sánchez-Ruiz, Antonio; Hevener, Kirk E; Narayanan, Ramesh; Clemons, William M Jr; Sarabia, Francisco; Kurosu, Michio

Role of TGF-β in pancreatic ductal adenocarcinoma progression and PD-L1 expression.

TGF-β在胰腺导管腺癌进展和PD-L1表达中的作用。

Hussain S Mazher, Kansal Rita G, Alvarez Marcus A, Hollingsworth T J, Elahi Abul, Miranda-Carboni Gustavo, Hendrick Leah E, Pingili Ajeeth K, Albritton Lorraine M, Dickson Paxton V, Deneve Jeremiah L, Yakoub Danny, Hayes D Neil, Kurosu Michio, Shibata David, Makowski Liza, Glazer Evan S

Substrate Tolerance of Bacterial Glycosyltransferase MurG: Novel Fluorescence-Based Assays

细菌糖基转移酶 MurG 的底物耐受性:新型荧光检测方法

Mitachi, Katsuhiko; Yun, Hyun Gi; Gillman, Cody D; Skorupinska-Tudek, Karolina; Swiezewska, Ewa; Clemons, William M Jr; Kurosu, Michio

Application of Mycobacterium smegmatis as a surrogate to evaluate drug leads against Mycobacterium tuberculosis

利用耻垢分枝杆菌作为替代菌株评价抗结核分枝杆菌的先导药物

Lelovic, Nada; Mitachi, Katsuhiko; Yang, Junshu; Lemieux, Maddie R; Ji, Yinduo; Kurosu, Michio

Semisynthesis of an Anticancer DPAGT1 Inhibitor from a Muraymycin Biosynthetic Intermediate

由穆拉霉素生物合成中间体半合成抗癌DPAGT1抑制剂

Mitachi, Katsuhiko; Kurosu, Shou M; Eslamimehr, Shakiba; Lemieux, Maddie R; Ishizaki, Yoshimasa; Clemons, William M Jr; Kurosu, Michio

Structure-based drug discovery by targeting N-glycan biosynthesis, dolichyl-phosphate N-acetylglucosaminephosphotransferase

通过靶向 N-糖生物合成、多萜磷酸 N-乙酰氨基葡萄糖磷酸转移酶进行基于结构的药物发现

Kurosu, Michio