A GIPR antagonist conjugated to GLP-1 analogues promotes weight loss with improved metabolic parameters in preclinical and phase 1 settings
在临床前和 I 期临床试验中,与 GLP-1 类似物偶联的 GIPR 拮抗剂可促进体重减轻并改善代谢指标。
期刊:Nature Metabolism
影响因子:20.8
doi:10.1038/s42255-023-00966-w
Véniant, Murielle M; Lu, Shu-Chen; Atangan, Larissa; Komorowski, Renee; Stanislaus, Shanaka; Cheng, Yuan; Wu, Bin; Falsey, James R; Hager, Todd; Thomas, Veena A; Ambhaikar, Malhar; Sharpsten, Lucie; Zhu, Yineng; Kurra, Vamsi; Jeswani, Rohini; Oberoi, Rajneet K; Parnes, Jane R; Honarpour, Narimon; Neutel, Joel; Strande, Jennifer L