日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Trophectoderm cell failure leads to peri-implantation lethality in Trpm7-deficient mouse embryos

滋养外胚层细胞衰竭导致Trpm7缺陷小鼠胚胎植入前死亡

Aline Schütz, Christin Richter, Petra Weissgerber, Volodymyr Tsvilovskyy, Michael Hesse, Roger Ottenheijm, Frank Zimmermann, Stefanie Buchholz, Rebekka Medert, Sascha Dlugosz, Vladimir Kuryshev, Vladimir Benes, Veit Flockerzi, Bernd K Fleischmann, Adolfo Cavalié, Marc Freichel

Efficacy and Safety of Netakimab, A Novel Anti-IL-17 Monoclonal Antibody, in Patients with Moderate to Severe Plaque Psoriasis. Results of A 54-Week Randomized Double-Blind Placebo-Controlled PLANETA Clinical Trial

Netakimab(一种新型抗IL-17单克隆抗体)治疗中重度斑块状银屑病患者的疗效和安全性:一项为期54周的随机、双盲、安慰剂对照PLANETA临床试验的结果

Puig, Luís; Bakulev, Andrey L; Kokhan, Muza M; Samtsov, Alexey V; Khairutdinov, Vladislav R; Morozova, Maria A; Zolkin, Nikita A; Kuryshev, Ivan V; Petrov, Alexey N; Artemeva, Antonina V; Zinkina-Orikhan, Arina V

Applying the CiPA approach to evaluate cardiac proarrhythmia risk of some antimalarials used off-label in the first wave of COVID-19

应用CiPA方法评估一些在COVID-19第一波疫情期间超适应症使用抗疟药的心脏致心律失常风险

Delaunois, Annie; Abernathy, Matthew; Anderson, Warren D; Beattie, Kylie A; Chaudhary, Khuram W; Coulot, Julie; Gryshkova, Vitalina; Hebeisen, Simon; Holbrook, Mark; Kramer, James; Kuryshev, Yuri; Leishman, Derek; Lushbough, Isabel; Passini, Elisa; Redfern, Will S; Rodriguez, Blanca; Rossman, Eric I; Trovato, Cristian; Wu, Caiyun; Valentin, Jean-Pierre

Development and validation of a potent and specific inhibitor for the CLC-2 chloride channel

开发和验证一种高效且特异性的CLC-2氯离子通道抑制剂

Koster, Anna K; Reese, Austin L; Kuryshev, Yuri; Wen, Xianlan; McKiernan, Keri A; Gray, Erin E; Wu, Caiyun; Huguenard, John R; Maduke, Merritt; Du Bois, J

Contribution of NAADP to Glutamate-Evoked Changes in Ca2+ Homeostasis in Mouse Hippocampal Neurons

NAADP 对小鼠海马神经元中谷氨酸诱发的 Ca2+ 稳态变化的贡献

Julia Hermann, Melanie Bender, Dagmar Schumacher, Marcel S Woo, Artem Shaposhnykov, Sina C Rosenkranz, Vladimir Kuryshev, Chris Meier, Andreas H Guse, Manuel A Friese, Marc Freichel, Volodymyr Tsvilovskyy

Corrigendum to "A systematic strategy for estimating hERG block potency and its implications in a new cardiac safety paradigm" [Toxicology and Applied Pharmacology volume 394C (2020) 114961]

对“评估 hERG 阻滞效力的系统策略及其在新的心脏安全范式中的意义”的更正[毒理学和应用药理学卷 394C (2020) 114961]

Ridder, Bradley J; Leishman, Derek J; Bridgland-Taylor, Matthew; Samieegohar, Mohammadreza; Han, Xiaomei; Wu, Wendy W; Randolph, Aaron; Tran, Phu; Sheng, Jiansong; Danker, Timm; Lindqvist, Anders; Konrad, Daniel; Hebeisen, Simon; Polonchuk, Liudmila; Gissinger, Evgenia; Renganathan, Muthukrishnan; Koci, Bryan; Wei, Haiyang; Fan, Jingsong; Levesque, Paul; Kwagh, Jae; Imredy, John; Zhai, Jin; Rogers, Marc; Humphries, Edward; Kirby, Robert; Stoelzle-Feix, Sonja; Brinkwirth, Nina; Rotordam, Maria Giustina; Becker, Nadine; Friis, Søren; Rapedius, Markus; Goetze, Tom A; Strassmaier, Tim; Okeyo, George; Kramer, James; Kuryshev, Yuri; Wu, Caiyun; Himmel, Herbert; Mirams, Gary R; Strauss, David G; Bardenet, Remi; Li, Zhihua

A systematic strategy for estimating hERG block potency and its implications in a new cardiac safety paradigm.

评估 hERG 阻滞效力的系统策略及其在新心脏安全范式中的意义

Ridder Bradley J, Leishman Derek J, Bridgland-Taylor Matthew, Samieegohar Mohammadreza, Han Xiaomei, Wu Wendy W, Randolph Aaron, Tran Phu, Sheng Jiansong, Danker Timm, Lindqvist Anders, Konrad Daniel, Hebeisen Simon, Polonchuk Liudmila, Gissinger Evgenia, Renganathan Muthukrishnan, Koci Bryan, Wei Haiyang, Fan Jingsong, Levesque Paul, Kwagh Jae, Imredy John, Zhai Jin, Rogers Marc, Humphries Edward, Kirby Robert, Stoelzle-Feix Sonja, Brinkwirth Nina, Rotordam Maria Giustina, Becker Nadine, Friis Søren, Rapedius Markus, Goetze Tom A, Strassmaier Tim, Okeyo George, Kramer James, Kuryshev Yuri, Wu Caiyun, Himmel Herbert, Mirams Gary R, Strauss David G, Bardenet Rémi, Li Zhihua

Assessment of an In Silico Mechanistic Model for Proarrhythmia Risk Prediction Under the CiPA Initiative

在CiPA计划下评估用于预测心律失常风险的计算机模拟机制模型

Li, Zhihua; Ridder, Bradley J; Han, Xiaomei; Wu, Wendy W; Sheng, Jiansong; Tran, Phu N; Wu, Min; Randolph, Aaron; Johnstone, Ross H; Mirams, Gary R; Kuryshev, Yuri; Kramer, James; Wu, Caiyun; Crumb, William J Jr; Strauss, David G

Pyrethroid neurotoxicity studies with bifenthrin indicate a mixed Type I/II mode of action

拟除虫菊酯类杀虫剂与联苯菊酯的神经毒性研究表明,其作用机制为I/II型混合型。

Gammon, Derek W; Liu, Zhiwei; Chandrasekaran, Appavu; El-Naggar, Shaaban F; Kuryshev, Yuri A; Jackson, Sharon

Molecular Evolution of Early-Onset Prostate Cancer Identifies Molecular Risk Markers and Clinical Trajectories

早期前列腺癌的分子演化揭示分子风险标志物和临床轨迹

Clarissa Gerhauser ,Francesco Favero ,Thomas Risch ,Ronald Simon ,Lars Feuerbach ,Yassen Assenov ,Doreen Heckmann ,Nikos Sidiropoulos ,Sebastian M Waszak ,Daniel Hübschmann ,Alfonso Urbanucci ,Etsehiwot G Girma ,Vladimir Kuryshev ,Leszek J Klimczak ,Natalie Saini ,Adrian M Stütz ,Dieter Weichenhan ,Lisa-Marie Böttcher ,Reka Toth ,Josephine D Hendriksen ,Christina Koop ,Pavlo Lutsik ,Sören Matzk ,Hans-Jörg Warnatz ,Vyacheslav Amstislavskiy ,Clarissa Feuerstein ,Benjamin Raeder ,Olga Bogatyrova ,Eva-Maria Schmitz ,Claudia Hube-Magg ,Martina Kluth ,Hartwig Huland ,Markus Graefen ,Chris Lawerenz ,Gervaise H Henry ,Takafumi N Yamaguchi ,Alicia Malewska ,Jan Meiners ,Daniela Schilling ,Eva Reisinger ,Roland Eils ,Matthias Schlesner ,Douglas W Strand ,Robert G Bristow ,Paul C Boutros ,Christof von Kalle ,Dmitry Gordenin ,Holger Sültmann ,Benedikt Brors ,Guido Sauter ,Christoph Plass ,Marie-Laure Yaspo ,Jan O Korbel ,Thorsten Schlomm ,Joachim Weischenfeldt