日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

GLP-1R/GCGR dual agonism dissipates hepatic steatosis to restore insulin sensitivity and rescue pancreatic β-cell function in obese male mice.

GLP-1R/GCGR 双重激动剂可消除肝脏脂肪变性,恢复肥胖雄性小鼠的胰岛素敏感性并挽救胰腺β细胞功能

Laker Rhianna C, Egolf Shaun, Will Sarah, Lantier Louise, McGuinness Owen P, Brown Charles, Bhagroo Nicholas, Oldham Stephanie, Kuszpit Kyle, Alfaro Alex, Li Xidan, Kang Taewook, Pellegrini Giovanni, Andréasson Anne-Christine, Kajani Sarina, Sitaula Sadichha, Larsen Martin R, Rhodes Christopher J

Characterization of PF-6142, a Novel, Non-Catecholamine Dopamine Receptor D1 Agonist, in Murine and Nonhuman Primate Models of Dopaminergic Activation

在小鼠和非人灵长类动物多巴胺能激活模型中对新型非儿茶酚胺多巴胺受体D1激动剂PF-6142进行表征

Rouba Kozak ,Tamás Kiss ,Keith Dlugolenski ,David E Johnson ,Roxanne R Gorczyca ,Kyle Kuszpit ,Brian D Harvey ,Polina Stolyar ,Stacey J Sukoff Rizzo ,William E Hoffmann ,Dmitri Volfson ,Mihaly Hajós ,Jennifer E Davoren ,Amanda L Abbott ,Graham V Williams ,Stacy A Castner ,David L Gray

Bioengineering of bacterial pathogens for noninvasive imaging and in vivo evaluation of therapeutics

利用生物工程技术改造细菌病原体,用于非侵入性成像和体内治疗效果评估

Rajamani, Sathish; Kuszpit, Kyle; Scarff, Jennifer M; Lundh, Linnea; Khan, Maisha; Brown, Jennifer; Stafford, Robert; Cazares, Lisa H; Panchal, Rekha G; Bocan, Thomas

[18F]DPA-714 PET Imaging Reveals Global Neuroinflammation in Zika Virus-Infected Mice

[18F]DPA-714 PET 成像揭示寨卡病毒感染小鼠的全身神经炎症

Kyle Kuszpit, Bradley S Hollidge, Xiankun Zeng, Robert G Stafford, Sharon Daye, Xiang Zhang, Falguni Basuli, Joseph W Golden, Rolf E Swenson, Darci R Smith, Thomas M Bocan

Neuropathogenesis of Zika Virus in a Highly Susceptible Immunocompetent Mouse Model after Antibody Blockade of Type I Interferon

干扰素 I 型抗体阻断后寨卡病毒在高度易感免疫功能正常小鼠模型中的神经发病机制

Darci R Smith, Bradley Hollidge, Sharon Daye, Xiankun Zeng, Candace Blancett, Kyle Kuszpit, Thomas Bocan, Jeff W Koehler, Susan Coyne, Tim Minogue, Tara Kenny, Xiaoli Chi, Soojin Yim, Lynn Miller, Connie Schmaljohn, Sina Bavari, Joseph W Golden

Inhibition of the human proteasome by imidazoline scaffolds

咪唑啉支架对人类蛋白酶体的抑制

Lauren M Azevedo, Theresa A Lansdell, Jacob R Ludwig, Robert A Mosey, Daljinder K Woloch, Dillon P Cogan, Gregory P Patten, Michael R Kuszpit, Jason S Fisk, Jetze J Tepe

The synthesis and in vivo evaluation of [18F]PF-9811: a novel PET ligand for imaging brain fatty acid amide hydrolase (FAAH)

[18F]PF-9811 的合成及体内评价:一种用于脑脂肪酸酰胺水解酶 (FAAH) 成像的新型 PET 配体

Skaddan, Marc B; Zhang, Lei; Johnson, Douglas S; Zhu, Aijun; Zasadny, Kenneth R; Coelho, Richard V; Kuszpit, Kyle; Currier, Gwen; Fan, Kuo-Hsien; Beck, Elizabeth M; Chen, Laigao; Drozda, Susan E; Balan, Gayatri; Niphakis, Micah; Cravatt, Benjamin F; Ahn, Kay; Bocan, Thomas; Villalobos, Anabella

PF-00477736 mediates checkpoint kinase 1 signaling pathway and potentiates docetaxel-induced efficacy in xenografts

PF-00477736 介导检查点激酶 1 信号通路并增强多西他赛在异种移植中诱导的疗效

Cathy Zhang, Zhengming Yan, Cory L Painter, Qin Zhang, Enhong Chen, Maria E Arango, Kyle Kuszpit, Kenneth Zasadny, Max Hallin, Jill Hallin, Anthony Wong, Dana Buckman, Guizhen Sun, Ming Qiu, Kenna Anderes, James G Christensen

Proton and sodium MRI assessment of emerging tumor chemotherapeutic resistance

利用质子和钠磁共振成像评估肿瘤化疗耐药性的出现

Schepkin, Victor D; Lee, Kuei C; Kuszpit, Kyle; Muthuswami, Mukilan; Johnson, Timothy D; Chenevert, Thomas L; Rehemtulla, Alnawaz; Ross, Brian D