日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Oxadiargyl analogs as potent inhibitors of Toxoplasma gondii protoporphyrinogen oxidase

氧二亚胺类似物是弓形虫原卟啉原氧化酶的强效抑制剂

Kwain, Samuel; Awasthi, Vikky; Islam, Rajib; Kore, Shivani; Polaski, Emma; Rees, Kerrick C; Dou, Zhicheng; Whitehead, Daniel C

Toward the clinical translation of safe intravenous long circulating ILNEs contrast agent for CT imaging

迈向安全有效的长循环静脉注射ILNEs造影剂在CT成像中的临床转化

Attia, Mohamed F; Marasco, Ryan N; Kwain, Samuel; Foxx, Charity; Whitehead, Daniel C; Kabanov, Alexander; Lee, Yueh Z

Assessment of the structure-activity relationship of analogs of the Naegleria fowleri enolase inhibitor HEX.

评估福氏耐格里阿米巴烯醇化酶抑制剂 HEX 类似物的构效关系

Kwain Samuel, Morris James W D, McKeon Jillian E M, Roster Colm P, Noori Monireh, Gibbs Aysiah R, Stevenson Iii Robert L, McMillen Colin D, Dominy Brian N, Morris James C, Whitehead Daniel C

Glucose metabolism in the pathogenic free-living amoebae: Tempting targets for treatment development

致病性自由生活变形虫的葡萄糖代谢:极具吸引力的治疗研发靶点

Milanes, Jillian E; Kwain, Samuel; Drawdy, Allyson; Dodson, Laura; Monaghan, Matthew T; Rice, Christopher A; Dominy, Brian N; Whitehead, Daniel C; Morris, James C

A cathepsin C-like protease mediates the post-translation modification of Toxoplasma gondii secretory proteins for optimal invasion and egress

一种类似组织蛋白酶C的蛋白酶介导弓形虫分泌蛋白的翻译后修饰,从而优化其入侵和释放。

Thornton, L Brock; Key, Melanie; Micchelli, Chiara; Stasic, Andrew J; Kwain, Samuel; Floyd, Katherine; Moreno, Silvia N J; Dominy, Brian N; Whitehead, Daniel C; Dou, Zhicheng

Enolase Inhibitors as Early Lead Therapeutics against Trypanosoma brucei

烯醇化酶抑制剂作为对抗布氏锥虫的早期先导疗法

Roster, Colm P; LaVigne, Danielle; Milanes, Jillian E; Knight, Emily; Anderson, Heidi D; Pizarro, Sabrina; Harding, Elijah M; Morris, Meredith T; Yan, Victoria C; Pham, Cong-Dat; Muller, Florian; Kwain, Samuel; Rees, Kerrick C; Dominy, Brian; Whitehead, Daniel C; Uddin, Md Nasir; Millward, Steven W; Morris, James C

A cathepsin C-like protease post-translationally modifies Toxoplasma gondii secretory proteins for optimal invasion and egress

一种类似组织蛋白酶C的蛋白酶对弓形虫分泌蛋白进行翻译后修饰,以优化其入侵和释放。

Thornton, L Brock; Key, Melanie; Micchelli, Chiara; Stasic, Andrew J; Kwain, Samuel; Floyd, Katherine; Moreno, Silvia N J; Dominy, Brian N; Whitehead, Daniel C; Dou, Zhicheng

In vitro effects and mechanisms of action of Bidens pilosa in Trypanosoma brucei

鬼针草对布氏锥虫的体外作用及其作用机制

Dofuor, Aboagye Kwarteng; Djameh, Georgina Isabella; Amoa-Bosompem, Michael; Kwain, Samuel; Osei, Enoch; Tetevi, Gilbert Mawuli; Ayertey, Frederick; Bolah, Peter; Okine, Laud Kenneth; Kyeremeh, Kwaku; Gwira, Theresa Manful; Ohashi, Mitsuko

Paenidigyamycin A, Potent Antiparasitic Imidazole Alkaloid from the Ghanaian Paenibacillus sp. DE2SH

帕尼迪吉霉素A,一种来自加纳帕尼芽孢杆菌属DE2SH菌株的强效抗寄生虫咪唑生物碱

Osei, Enoch; Kwain, Samuel; Mawuli, Gilbert Tetevi; Anang, Abraham Kwabena; Owusu, Kofi Baffour-Awuah; Camas, Mustafa; Camas, Anil Sazak; Ohashi, Mitsuko; Alexandru-Crivac, Cristina-Nicoleta; Deng, Hai; Jaspars, Marcel; Kyeremeh, Kwaku