日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

High throughput quantitative tracking of Plasmodium falciparum clonal blood stage parasite growth and applications for antimalarial drug discovery

高通量定量追踪恶性疟原虫克隆血期寄生虫的生长及其在抗疟药物发现中的应用

Cheng, Zhe; Ru, Liyang; Hoang, Andrew; Wang, Mingyu; Ganjikunta, Suryanarayana; Maher, Steven P; Kyle, Dennis E

A drug repurposing approach reveals targetable epigenetic pathways in Plasmodium vivax hypnozoites.

药物再利用方法揭示了间日疟原虫休眠子中可靶向的表观遗传通路

Maher Steven P, Bakowski Malina A, Vantaux Amélie, Flannery Erika L, Andolina Chiara, Gupta Mohit, Antonova-Koch Yevgeniya, Argomaniz Magdalena, Cabrera-Mora Monica, Campo Brice, Chao Alexander T, Chatterjee Arnab K, Cheng Wayne T, Chuenchob Vorada, Cooper Caitlin A, Cottier Karissa, Galinski Mary R, Harupa-Chung Anke, Ji Hana, Joseph Sean B, Lenz Todd, Lonardi Stefano, Matheson Jessica, Mikolajczak Sebastian A, Moeller Timothy, Orban Agnes, Padín-Irizarry Vivian, Pan Kastin, Péneau Julie, Prudhomme Jacques, Roesch Camille, Ruberto Anthony, Sabnis Saniya S, Saney Celia L, Sattabongkot Jetsumon, Sereshki Saleh, Suriyakan Sangrawee, Ubalee Ratawan, Wang Yinsheng, Wasisakun Praphan, Yin Jiekai, Popovici Jean, McNamara Case W, Joyner Chester, Nosten François H, Witkowski Benoît, Le Roch Karine G, Kyle Dennis E

Characterization of β-Carboline Derivatives Reveals a High Barrier to Resistance and Potent Activity against Ring-Stage and DHA-Induced Dormant Plasmodium falciparum

β-咔啉衍生物的表征揭示了其对环状体和DHA诱导的休眠期恶性疟原虫具有高抗药性屏障和强效活性。

Haney, Reagan S; Butler, Joshua H; Wardlaw, Lyric A; Merino, Emilio F; Mendiola, Victoria; Cooper, Caitlin A; Mathew, Jopaul; Tumwebaze, Patrick K; Rosenthal, Philip J; Cooper, Roland A; Kyle, Dennis E; Rizopoulos, Zaira; Baud, Delphine; Brand, Stephen; Totrov, Maxim; Carlier, Paul R; Cassera, Maria Belen

Virulence of Naegleria fowleri isolates varies significantly in the mouse model of primary amoebic meningoencephalitis

在原发性阿米巴脑膜脑炎小鼠模型中,福氏耐格里阿米巴分离株的毒力差异显著。

Russell, A Cassiopeia; Schiff, Erica; Dainis, Joseph; Jones, Håkon; Rice, Christopher A; Kyle, Dennis E

Secreted small RNAs of Naegleria fowleri are biomarkers for diagnosis of primary amoebic meningoencephalitis

福氏耐格里阿米巴分泌的小RNA是原发性阿米巴脑膜脑炎的诊断生物标志物。

Russell, A Cassiopeia; Dainis, Joseph; Alexander, Jose; Ali, Ibne Karim M; Kyle, Dennis E

Optimization of diastereomeric dihydropyridines as antimalarials

优化非对映异构二氢吡啶类化合物作为抗疟药

Van Horn, Kurt S; Zhao, Yingzhao; Parvatkar, Prakash T; Maier, Julie; Mutka, Tina; Lacrue, Alexis; Brockmeier, Fabian; Ebert, Daniel; Wu, Wesley; Casandra, Debora R; Namelikonda, Niranjan; Yacoub, Jeanine; Sigal, Martina; Knapp, Spencer; Floyd, David; Waterson, David; Burrows, Jeremy N; Duffy, James; DeRisi, Joseph L; Kyle, Dennis E; Guy, R Kiplin; Manetsch, Roman

Extended blood stage sensitivity profiles of Plasmodium cynomolgi to doxycycline and tafenoquine, as a model for Plasmodium vivax.

以猴疟原虫血液期对多西环素和他非诺喹的敏感性谱为例,研究间日疟原虫

Christensen Peter, Cinzah Rosy, Suwanarusk Rossarin, Chua Adeline Chiew Yen, Kaneko Osamu, Kyle Dennis E, Aung Htin Lin, Matheson Jessica, Bifani Pablo, Rénia Laurent, Cook Gregory M, Snounou Georges, Russell Bruce

In Vitro Antimalarial Activity of Trichothecenes against Liver and Blood Stages of Plasmodium Species

体外抗疟活性研究表明,单端孢霉烯族化合物对疟原虫肝期和血期均具有抗疟活性

Parvatkar, Prakash T; Maher, Steven P; Zhao, Yingzhao; Cooper, Caitlin A; de Castro, Sagan T; Péneau, Julie; Vantaux, Amélie; Witkowski, Benoît; Kyle, Dennis E; Manetsch, Roman

The influence of oviposition status on measures of transmission potential in malaria-infected mosquitoes depends on sugar availability

产卵状态对疟疾感染蚊子传播潜力的影响取决于糖的供应情况。

Shiau, Justine C; Garcia-Diaz, Nathan; Kyle, Dennis E; Pathak, Ashutosh K

Type-I IFNs induce GBPs and lysosomal defense in hepatocytes to control malaria

I型干扰素诱导肝细胞中糖蛋白结合蛋白(GBP)和溶酶体防御机制,从而控制疟疾。

Marques-da-Silva, Camila; Schmidt-Silva, Clyde; Bowers, Carson; Charles-Chess, Essel; Shiau, Justine C; Park, Eui-Soon; Yuan, Zhongyu; Kim, Bae-Hoon; Kyle, Dennis E; Harty, John T; MacMicking, John D; Kurup, Samarchith P