Myosin modulator Aficamten inhibits force in cardiac muscle by altering myosin's biochemical activity without changing thick filament structure
肌球蛋白调节剂阿菲卡明通过改变肌球蛋白的生化活性来抑制心肌收缩力,而不改变粗肌丝的结构。
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doi:10.1101/2025.05.14.654110
Mohran, Saffie; Kooiker, Kristina B; Naim, Ateeqa; Pilagov, Matvey; Asencio, Anthony; Turner, Kyrah L; Ma, Weikang; Flint, Galina; Jiang, Siyao; Zhao, Jing; McMillen, Timothy S; Mandrycky, Christian; Mahoney-Schaefer, Max; Irving, Thomas C; Tanner, Bertrand C W; Kad, Neil M; Regnier, Michael; Moussavi-Harami, Farid