Discovery of a PDE4B and PDE4D selective bifunctional degrader for management of chronic inflammatory disorders.
发现一种对PDE4B和PDE4D具有选择性的双功能降解剂,用于治疗慢性炎症性疾病。
期刊:Journal of Translational Autoimmunity
影响因子:3.6
doi:10.1016/j.jtauto.2025.100329
Shakya Arvind, Liu Qiao, Lai Chon, Baker Sherry, Greene Steven, Erdman Paul, Rathnayake Athri, Schoolmeesters Angela, Blair Connor M, Kyurkchieva Elka, Rajapakse Navin, Lam Imelda, Sin Yuan Yan, Baillie George S, Huang Shenlin, Chourasia Aparajita H, Fung Leah