日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A novel approach for modeling in vivo enzyme turnover in the presence of a suicide inhibitor drug: A proof-of-concept brain PET study on MAG lipase

一种模拟体内酶周转(在自杀性抑制剂药物存在下)的新方法:MAG脂肪酶的脑PET概念验证研究

Volpi, Tommaso; Holden, Daniel; Gallezot, Jean-Dominique; Nabulsi, Nabeel; Lim, Keunpoong; Labaree, David; Gao, Hong; Kapinos, Michael; Keliher, Edmund J; Fonseca, Kari R; Trapa, Patrick; Varrone, Andrea; Halldin, Christer; Maresca, Kevin P; Huang, Yiyun; Carson, Richard E

First-in-Human Assessment of (11)C-LSN3172176, an M1 Muscarinic Acetylcholine Receptor PET Radiotracer

首次人体评估 (11)C-LSN3172176,一种 M1 毒蕈碱乙酰胆碱受体 PET 放射性示踪剂

Naganawa, Mika; Nabulsi, Nabeel; Henry, Shannan; Matuskey, David; Lin, Shu-Fei; Slieker, Lawrence; Schwarz, Adam J; Kant, Nancy; Jesudason, Cynthia; Ruley, Kevin; Navarro, Antonio; Gao, Hong; Ropchan, Jim; Labaree, David; Carson, Richard E; Huang, Yiyun

Separating dopamine D(2) and D(3) receptor sources of [(11)C]-(+)-PHNO binding potential: Independent component analysis of competitive binding

分离多巴胺 D(2) 和 D(3) 受体来源的 [(11)C]-(+)-PHNO 结合潜能:竞争性结合的独立成分分析

Smart, Kelly; Gallezot, Jean-Dominique; Nabulsi, Nabeel; Labaree, David; Zheng, Ming-Qiang; Huang, Yiyun; Carson, Richard E; Hillmer, Ansel T; Worhunsky, Patrick D

Body Mass Index and Age Effects on Brain 11β-Hydroxysteroid Dehydrogenase Type 1: a Positron Emission Tomography Study

体重指数和年龄对脑部11β-羟类固醇脱氢酶1型的影响:一项正电子发射断层扫描研究

Bini, Jason; Bhatt, Shivani; Hillmer, Ansel T; Gallezot, Jean-Dominique; Nabulsi, Nabeel; Pracitto, Richard; Labaree, David; Kapinos, Michael; Ropchan, Jim; Matuskey, David; Sherwin, Robert S; Jastreboff, Ania M; Carson, Richard E; Cosgrove, Kelly; Huang, Yiyun

Synthesis and in Vivo Evaluation of a Novel PET Radiotracer for Imaging of Synaptic Vesicle Glycoprotein 2A (SV2A) in Nonhuman Primates

新型 PET 放射性示踪剂的合成及体内评估,用于非人类灵长类动物突触囊泡糖蛋白 2A (SV2A) 成像

Songye Li, Zhengxin Cai, Xiaoai Wu, Daniel Holden, Richard Pracitto, Michael Kapinos, Hong Gao, David Labaree, Nabeel Nabulsi, Richard E Carson, Yiyun Huang

Binge alcohol use is not associated with alterations in striatal dopamine receptor binding or dopamine release

酗酒与纹状体多巴胺受体结合或多巴胺释放的改变无关

Wai, Jonathan M; Grassetti, Alexander; Slifstein, Mark; Matuskey, David; Nabulsi, Nabeel; Ropchan, Jim; Labaree, David; Huang, Yiyun; Martinez, Diana

Development and In Vivo Evaluation of a κ-Opioid Receptor Agonist as a PET Radiotracer with Superior Imaging Characteristics

开发并体内评价一种具有优异成像特性的κ-阿片受体激动剂作为PET放射性示踪剂

Li, Songye; Zheng, Ming-Qiang; Naganawa, Mika; Kim, Sujin; Gao, Hong; Kapinos, Michael; Labaree, David; Huang, Yiyun

Evaluation of Pancreatic VMAT2 Binding with Active and Inactive Enantiomers of [(18)F]FP-DTBZ in Healthy Subjects and Patients with Type 1 Diabetes

在健康受试者和1型糖尿病患者中评估[(18)F]FP-DTBZ活性和非活性对映体与胰腺VMAT2的结合情况

Naganawa, Mika; Lim, Keunpoong; Nabulsi, Nabeel B; Lin, Shu-Fei; Labaree, David; Ropchan, Jim; Herold, Kevan C; Huang, Yiyun; Harris, Paul; Ichise, Masanori; Cline, Gary W; Carson, Richard E

Novel (18)F-Labeled κ-Opioid Receptor Antagonist as PET Radiotracer: Synthesis and In Vivo Evaluation of (18)F-LY2459989 in Nonhuman Primates

新型 (18)F 标记的 κ-阿片受体拮抗剂作为 PET 放射性示踪剂:(18)F-LY2459989 在非人灵长类动物中的合成和体内评价

Li, Songye; Cai, Zhengxin; Zheng, Ming-Qiang; Holden, Daniel; Naganawa, Mika; Lin, Shu-Fei; Ropchan, Jim; Labaree, David; Kapinos, Michael; Lara-Jaime, Teresa; Navarro, Antonio; Huang, Yiyun

PET imaging of α(7) nicotinic acetylcholine receptors: a comparative study of [(18)F]ASEM and [(18)F]DBT-10 in nonhuman primates, and further evaluation of [(18)F]ASEM in humans

α(7)尼古丁乙酰胆碱受体的PET成像:非人灵长类动物中[(18)F]ASEM和[(18)F]DBT-10的比较研究,以及[(18)F]ASEM在人体中的进一步评估

Hillmer, Ansel T; Li, Songye; Zheng, Ming-Qiang; Scheunemann, Matthias; Lin, Shu-Fei; Nabulsi, Nabeel; Holden, Daniel; Pracitto, Richard; Labaree, David; Ropchan, Jim; Teodoro, Rodrigo; Deuther-Conrad, Winnie; Esterlis, Irina; Cosgrove, Kelly P; Brust, Peter; Carson, Richard E; Huang, Yiyun