An allosteric pan-TEAD inhibitor blocks oncogenic YAP/TAZ signaling and overcomes KRAS G12C inhibitor resistance
变构泛 TEAD 抑制剂阻断致癌 YAP/TAZ 信号传导并克服 KRAS G12C 抑制剂耐药性
期刊:Nature Cancer
影响因子:23.5
doi:10.1038/s43018-023-00577-0
Thijs J Hagenbeek #, Jason R Zbieg #, Marc Hafner #, Rana Mroue, Jennifer A Lacap, Nicole M Sodir, Cameron L Noland, Shervin Afghani, Ayush Kishore, Kamakoti P Bhat, Xiaosai Yao, Stephen Schmidt, Saundra Clausen, Micah Steffek, Wendy Lee, Paul Beroza, Scott Martin, Eva Lin, Rina Fong, Paola Di Lello