日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

CC48 a new CB2R agonist/FAAH inhibitor dual drug blocks gastric cancer progression and overcomes paclitaxel resistance.

CC48 是一种新型 CB2R 激动剂/FAAH 抑制剂双效药物,可阻断胃癌进展并克服紫杉醇耐药性

Schirizzi Annalisa, Renna Natasha, De Leonardis Giampiero, Montanaro Rosangela, Mastropasqua Francesco, Graziano Giovanni, Riganti Chiara, Pisano Isabella, Laghezza Antonio, Abate Carmen, Stefanachi Angela, Colabufo Nicola Antonio, Caccioppoli Cristina, Bianco Giusy, Valentini Anna Maria, Armentano Raffaele, Giannelli Gianluigi, Contino Marialessandra, D'Alessandro Rosalba

Deep Eutectic Solvents (DESs) as Alternative Sustainable Media for the Extraction and Characterization of Bioactive Compounds from Winemaking Industry Wastes.

深共熔溶剂(DES)作为替代可持续介质,用于从酿酒工业废料中提取和表征生物活性化合物

Roselli Vincenzo, Leuci Rosalba, Pugliese Gianluca, Barbarossa Alexia, Laghezza Antonio, Paparella Marco, Carocci Alessia, Tufarelli Vincenzo, Gambacorta Lucia, Piemontese Luca

AMALPHI: A Machine Learning Platform for Predicting Drug-Induced PhospholIpidosis

AMALPHI:用于预测药物诱导磷脂沉积症的机器学习平台

Lomuscio, Maria Cristina; Abate, Carmen; Alberga, Domenico; Laghezza, Antonio; Corriero, Nicola; Colabufo, Nicola Antonio; Saviano, Michele; Delre, Pietro; Mangiatordi, Giuseppe Felice

Bone-Seeking Matrix Metalloproteinase Inhibitors for the Treatment of Skeletal Malignancy

用于治疗骨骼恶性肿瘤的亲骨基质金属蛋白酶抑制剂

Laghezza, Antonio; Piemontese, Luca; Brunetti, Leonardo; Caradonna, Alessia; Agamennone, Mariangela; Di Pizio, Antonella; Pochetti, Giorgio; Montanari, Roberta; Capelli, Davide; Tauro, Marilena; Loiodice, Fulvio; Tortorella, Paolo

Single-Nucleotide Polymorphism of PPARγ, a Protein at the Crossroads of Physiological and Pathological Processes

PPARγ单核苷酸多态性:一种处于生理和病理过程交汇点的蛋白质

Petrosino, Maria; Lori, Laura; Pasquo, Alessandra; Lori, Clorinda; Consalvi, Valerio; Minicozzi, Velia; Morante, Silvia; Laghezza, Antonio; Giorgi, Alessandra; Capelli, Davide; Chiaraluce, Roberta

Betulinic acid is a PPARγ antagonist that improves glucose uptake, promotes osteogenesis and inhibits adipogenesis

桦木酸是一种PPARγ拮抗剂,可改善葡萄糖摄取、促进骨生成并抑制脂肪生成。

Brusotti, Gloria; Montanari, Roberta; Capelli, Davide; Cattaneo, Giulia; Laghezza, Antonio; Tortorella, Paolo; Loiodice, Fulvio; Peiretti, Franck; Bonardo, Bernadette; Paiardini, Alessandro; Calleri, Enrica; Pochetti, Giorgio

Seeking for Non-Zinc-Binding MMP-2 Inhibitors: Synthesis, Biological Evaluation and Molecular Modelling Studies

寻找非锌结合型MMP-2抑制剂:合成、生物学评价和分子建模研究

Ammazzalorso, Alessandra; De Filippis, Barbara; Campestre, Cristina; Laghezza, Antonio; Marrone, Alessandro; Amoroso, Rosa; Tortorella, Paolo; Agamennone, Mariangela

Insights into the complex formed by matrix metalloproteinase-2 and alloxan inhibitors: molecular dynamics simulations and free energy calculations

基质金属蛋白酶-2与阿洛沙抑制剂形成的复合物的研究进展:分子动力学模拟和自由能计算

Giangreco, Ilenia; Lattanzi, Gianluca; Nicolotti, Orazio; Catto, Marco; Laghezza, Antonio; Leonetti, Francesco; Stefanachi, Angela; Carotti, Angelo