日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Cyclohexyl-griselimycin Is Active against Mycobacterium abscessus in Mice

环己基-格里西利霉素对小鼠脓肿分枝杆菌有效

Aragaw, Wassihun Wedajo; Roubert, Christine; Fontaine, Evelyne; Lagrange, Sophie; Zimmerman, Matthew D; Dartois, Véronique; Gengenbacher, Martin; Dick, Thomas

Identification of β-Lactams Active against Mycobacterium tuberculosis by a Consortium of Pharmaceutical Companies and Academic Institutions

由制药公司和学术机构组成的联盟对抗结核分枝杆菌的β-内酰胺类抗生素进行鉴定

Gold, Ben; Zhang, Jun; Quezada, Landys Lopez; Roberts, Julia; Ling, Yan; Wood, Madeleine; Shinwari, Wasima; Goullieux, Laurent; Roubert, Christine; Fraisse, Laurent; Bacqué, Eric; Lagrange, Sophie; Filoche-Rommé, Bruno; Vieth, Michal; Hipskind, Philip A; Jungheim, Louis N; Aubé, Jeffrey; Scarry, Sarah M; McDonald, Stacey L; Li, Kelin; Perkowski, Andrew; Nguyen, Quyen; Dartois, Véronique; Zimmerman, Matthew; Olsen, David B; Young, Katherine; Bonnett, Shilah; Joerss, Douglas; Parish, Tanya; Boshoff, Helena I; Arora, Kriti; Barry, Clifton E 3rd; Guijarro, Laura; Anca, Sara; Rullas, Joaquín; Rodríguez-Salguero, Beatriz; Martínez-Martínez, Maria S; Porras-De Francisco, Esther; Cacho, Monica; Barros-Aguirre, David; Smith, Paul; Berthel, Steven J; Nathan, Carl; Bates, Robert H

N-Acetylglucosamine-1-Phosphate Transferase, WecA, as a Validated Drug Target in Mycobacterium tuberculosis

N-乙酰氨基葡萄糖-1-磷酸转移酶 WecA 是结核分枝杆菌中已验证的药物靶点

Huszár, Stanislav; Singh, Vinayak; Polčicová, Alica; Baráth, Peter; Barrio, María Belén; Lagrange, Sophie; Leblanc, Véronique; Nacy, Carol A; Mizrahi, Valerie; Mikušová, Katarína

The Inosine Monophosphate Dehydrogenase, GuaB2, Is a Vulnerable New Bactericidal Drug Target for Tuberculosis

肌苷单磷酸脱氢酶 GuaB2 是结核病新型杀菌药物的易损靶点

Singh, Vinayak; Donini, Stefano; Pacitto, Angela; Sala, Claudia; Hartkoorn, Ruben C; Dhar, Neeraj; Keri, Gyorgy; Ascher, David B; Mondésert, Guillaume; Vocat, Anthony; Lupien, Andréanne; Sommer, Raphael; Vermet, Hélène; Lagrange, Sophie; Buechler, Joe; Warner, Digby F; McKinney, John D; Pato, Janos; Cole, Stewart T; Blundell, Tom L; Rizzi, Menico; Mizrahi, Valerie

A trisubstituted benzimidazole cell division inhibitor with efficacy against Mycobacterium tuberculosis.

一种对结核分枝杆菌有效的三取代苯并咪唑细胞分裂抑制剂

Knudson Susan E, Awasthi Divya, Kumar Kunal, Carreau Alexandra, Goullieux Laurent, Lagrange Sophie, Vermet Hélèn, Ojima Iwao, Slayden Richard A