日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Distinct oligomeric assemblies of STING induced by non-nucleotide agonists.

非核苷酸激动剂诱导的 STING 的不同寡聚体组装体

Gharpure Anant, Sulpizio Ariana, Loeffler Johannes R, Fernández-Quintero Monica L, Tran Andy S, Lairson Luke L, Ward Andrew B

Insights into Free Drug Release from Efficacious N-Acyl O-Aminophenol Duocarmycin Prodrugs.

对高效N-酰基O-氨基苯酚杜卡霉素前药的游离药物释放的深入研究

Chakraborty Nilanjana, Momirov Jelena, Radakovic Aleksandar, Chatterjee Shreyosree, Kirchhoff Aaron M, Kolb Anna-Lena, West Thomas J, Sanchez Brittany B, Martinez-Bartolome Salvador, Saviola Anthony, McClatchy Daniel, Yates John R 3rd, Chen Jason S, Lairson Luke L, Felding Brunie H, Boger Dale L

Induced cell phenotype activity recording of DNA-tagged ligands

DNA标记配体的诱导细胞表型活性记录

Sander, Philipp N; Gillen Miller, Jared T; Lairson, Luke L

Discovery of PLD4 modulators by high-throughput screening and kinetic analysis

通过高通量筛选和动力学分析发现PLD4调节剂

Lee, Jinny Claire; Shirey, Ryan J; Turner, Lewis D; Park, Hyeri; Lairson, Luke L; Janda, Kim D

A Cell Type Selective YM155 Prodrug Targets Receptor-Interacting Protein Kinase 2 to Induce Brain Cancer Cell Death

一种细胞类型选择性前药YM155靶向受体相互作用蛋白激酶2,诱导脑癌细胞死亡

West, Thomas J; Bi, Junfeng; Martínez-Peña, Francisco; Curtis, Ellis J; Gazaniga, Nathalia R; Mischel, Paul S; Lairson, Luke L

Optimization of 3-aminotetrahydrothiophene 1,1-dioxides with improved potency and efficacy as non-electrophilic antioxidant response element (ARE) activators

优化3-氨基四氢噻吩-1,1-二氧化物,以提高其作为非亲电抗氧化反应元件(ARE)激活剂的效力和功效

Jo, Jeyun; Kim, Jisu; Ibrahim, Lara; Kumar, Manoj; Iaconelli, Jonathan; Tran, Cong So; Moon, Hyung Ryong; Jung, Yunjin; Wiseman, R Luke; Lairson, Luke L; Chatterjee, Arnab K; Bollong, Michael J; Yun, Hwayoung

Discovery and optimization of aspartate aminotransferase 1 inhibitors to target redox balance in pancreatic ductal adenocarcinoma

发现和优化天冬氨酸氨基转移酶 1 抑制剂以靶向胰腺导管腺癌的氧化还原平衡

Anglin, Justin; Zavareh, Reza Beheshti; Sander, Philipp N; Haldar, Daniel; Mullarky, Edouard; Cantley, Lewis C; Kimmelman, Alec C; Lyssiotis, Costas A; Lairson, Luke L

Systems biology guided by XCMS Online metabolomics

系统生物学,以XCMS在线代谢组学为指导

Huan, Tao; Forsberg, Erica M; Rinehart, Duane; Johnson, Caroline H; Ivanisevic, Julijana; Benton, H Paul; Fang, Mingliang; Aisporna, Aries; Hilmers, Brian; Poole, Farris L; Thorgersen, Michael P; Adams, Michael W W; Krantz, Gregory; Fields, Matthew W; Robbins, Paul D; Niedernhofer, Laura J; Ideker, Trey; Majumder, Erica L; Wall, Judy D; Rattray, Nicholas J W; Goodacre, Royston; Lairson, Luke L; Siuzdak, Gary

Small molecule-mediated inhibition of myofibroblast transdifferentiation for the treatment of fibrosis

小分子介导的肌成纤维细胞转分化抑制治疗纤维化

Bollong, Michael J; Yang, Baiyuan; Vergani, Naja; Beyer, Brittney A; Chin, Emily N; Zambaldo, Claudio; Wang, Danling; Chatterjee, Arnab K; Lairson, Luke L; Schultz, Peter G

Mapping Protein Targets of Bioactive Small Molecules Using Lipid-Based Chemical Proteomics

利用基于脂质的化学蛋白质组学绘制生物活性小分子的蛋白质靶标图谱

Lum, Kenneth M; Sato, Yoshiaki; Beyer, Brittney A; Plaisted, Warren C; Anglin, Justin L; Lairson, Luke L; Cravatt, Benjamin F