日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Ion channel inhibition by targeted recruitment of NEDD4-2 with divalent nanobodies.

利用二价纳米抗体靶向募集 NEDD4-2 来抑制离子通道。

Darko-Boateng Arden, Afriyie Emmanuel, Morgenstern Travis J, Shanmugam Sri Karthika, Zou Xinle, Laloudakis Yianni D, Choudhury Papiya, Desai Meera, Kass Robert S, Vallese Francesca, Clarke Oliver B, Colecraft Henry M

Xanomeline displays concomitant orthosteric and allosteric binding modes at the M(4) mAChR

Xanomeline 在 M(4) mAChR 上表现出正构和变构结合模式。

Burger, Wessel A C; Pham, Vi; Vuckovic, Ziva; Powers, Alexander S; Mobbs, Jesse I; Laloudakis, Yianni; Glukhova, Alisa; Wootten, Denise; Tobin, Andrew B; Sexton, Patrick M; Paul, Steven M; Felder, Christian C; Danev, Radostin; Dror, Ron O; Christopoulos, Arthur; Valant, Celine; Thal, David M

Molecular mechanism of biased signaling at the kappa opioid receptor.

kappa阿片受体偏向性信号传导的分子机制

El Daibani Amal, Paggi Joseph M, Kim Kuglae, Laloudakis Yianni D, Popov Petr, Bernhard Sarah M, Krumm Brian E, Olsen Reid H J, Diberto Jeffrey, Carroll F Ivy, Katritch Vsevolod, Wünsch Bernhard, Dror Ron O, Che Tao

Author Correction: Structural basis of efficacy-driven ligand selectivity at GPCRs

作者更正:GPCR 上功效驱动配体选择性的结构基础

Powers, Alexander S; Pham, Vi; Burger, Wessel A C; Thompson, Geoff; Laloudakis, Yianni; Barnes, Nicholas W; Sexton, Patrick M; Paul, Steven M; Christopoulos, Arthur; Thal, David M; Felder, Christian C; Valant, Celine; Dror, Ron O

Selective posttranslational inhibition of CaVβ1-associated voltage-dependent calcium channels with a functionalized nanobody

利用功能化纳米抗体选择性翻译后抑制 CaVβ1 相关电压依赖性钙通道

Travis J Morgenstern, Neha Nirwan, Erick O Hernández-Ochoa, Hugo Bibollet, Papiya Choudhury, Yianni D Laloudakis, Manu Ben Johny, Roger A Bannister, Martin F Schneider, Daniel L Minor Jr, Henry M Colecraft

Biophysical characterization and a roadmap towards the NMR solution structure of G0S2, a key enzyme in non-alcoholic fatty liver disease

G0S2(非酒精性脂肪肝疾病中的关键酶)的生物物理表征及其核磁共振溶液结构解析路线图

Moran, Michael W; Ramirez, Elizabeth P; Zook, James D; Saarinen, Alicia M; Baravati, Bobby; Goode, Matthew R; Laloudakis, Vasiliki; Kaschner, Emily K; Olson, Tien L; Craciunescu, Felicia M; Hansen, Debra T; Liu, Jun; Fromme, Petra