Xanomeline displays concomitant orthosteric and allosteric binding modes at the M(4) mAChR
Xanomeline 在 M(4) mAChR 上表现出正构和变构结合模式。
期刊:Nature Communications
影响因子:15.7
doi:10.1038/s41467-023-41199-5
Burger, Wessel A C; Pham, Vi; Vuckovic, Ziva; Powers, Alexander S; Mobbs, Jesse I; Laloudakis, Yianni; Glukhova, Alisa; Wootten, Denise; Tobin, Andrew B; Sexton, Patrick M; Paul, Steven M; Felder, Christian C; Danev, Radostin; Dror, Ron O; Christopoulos, Arthur; Valant, Celine; Thal, David M