日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Sulphostin-inspired N-phosphonopiperidones as selective covalent DPP8 and DPP9 inhibitors.

受磺基膦酸酯启发而合成的 N-膦酸哌啶酮类化合物作为选择性共价 DPP8 和 DPP9 抑制剂

Sewald Leonard, Tabak Werner W A, Fehr Lorenz, Zolg Samuel, Najdzion Maja, Verhoef Carlo J A, Podlesainski David, Geiss-Friedlander Ruth, Lammens Alfred, Kaschani Farnusch, Hellerschmied Doris, Huber Robert, Kaiser Markus

The Discovery of Bridged Benzoazepine Amides as Selective Allosteric Modulators of RIPK1

桥联苯并氮杂卓酰胺作为RIPK1选择性变构调节剂的发现

Chen, Joanna L; Methot, Joey L; Mitcheltree, Matthew J; Musacchio, Andrew; Corcoran, Emily B; Feng, Guo; Lammens, Alfred; Maskos, Klaus; Palte, Rachel L; Rickard, Meredith M; Otte, Karin M; Mansueto, My S; Venkat, Sriraman; Sondey, Christopher; Thomsen, Maren; Lesburg, Charles A; Fradera, Xavier; Fell, Matthew J; DiMauro, Erin F; Siliphaivanh, Phieng

Structures, functions and adaptations of the human LINE-1 ORF2 protein

人类LINE-1 ORF2蛋白的结构、功能和适应性

Baldwin, Eric T; van Eeuwen, Trevor; Hoyos, David; Zalevsky, Arthur; Tchesnokov, Egor P; Sánchez, Roberto; Miller, Bryant D; Di Stefano, Luciano H; Ruiz, Francesc Xavier; Hancock, Matthew; Işik, Esin; Mendez-Dorantes, Carlos; Walpole, Thomas; Nichols, Charles; Wan, Paul; Riento, Kirsi; Halls-Kass, Rowan; Augustin, Martin; Lammens, Alfred; Jestel, Anja; Upla, Paula; Xibinaku, Kera; Congreve, Samantha; Hennink, Maximiliaan; Rogala, Kacper B; Schneider, Anna M; Fairman, Jennifer E; Christensen, Shawn M; Desrosiers, Brian; Bisacchi, Gregory S; Saunders, Oliver L; Hafeez, Nafeeza; Miao, Wenyan; Kapeller, Rosana; Zaller, Dennis M; Sali, Andrej; Weichenrieder, Oliver; Burns, Kathleen H; Götte, Matthias; Rout, Michael P; Arnold, Eddy; Greenbaum, Benjamin D; Romero, Donna L; LaCava, John; Taylor, Martin S

Utilization of Metabolite Identification and Structural Data to Guide Design of Low-Dose IDO1 Inhibitors

利用代谢物鉴定和结构数据指导低剂量IDO1抑制剂的设计

Hopkins, Brett; Zhang, Hongjun; Bharathan, Indu; Li, Derun; Pu, Qinglin; Zhou, Hua; Martinot, Theodore A; Fradera, Xavier; Lammens, Alfred; Lesburg, Charles A; Cohen, Ryan D; Ballard, Jeanine; Knemeyer, Ian; Otte, Karin; Vincent, Stella; Miller, J Richard; Solban, Nicolas; Cheng, Mangeng; Geda, Prasanthi; Smotrov, Nadya; Song, Xuelei; Bennett, David Jonathan; Han, Yongxin

Carbamate and N-Pyrimidine Mitigate Amide Hydrolysis: Structure-Based Drug Design of Tetrahydroquinoline IDO1 Inhibitors

氨基甲酸酯和N-嘧啶可减轻酰胺水解:基于结构的四氢喹啉IDO1抑制剂药物设计

Li, Derun; Deng, Yongqi; Achab, Abdelghani; Bharathan, Indu; Hopkins, Brett Andrew; Yu, Wensheng; Zhang, Hongjun; Sanyal, Sulagna; Pu, Qinglin; Zhou, Hua; Liu, Kun; Lim, Jongwon; Fradera, Xavier; Lesburg, Charles A; Lammens, Alfred; Martinot, Theodore A; Cohen, Ryan D; Doty, Amy C; Ferguson, Heidi; Nickbarg, Elliott B; Cheng, Mangeng; Spacciapoli, Peter; Geda, Prasanthi; Song, Xuelei; Smotrov, Nadya; Abeywickrema, Pravien; Andrews, Christine; Chamberlin, Chad; Mabrouk, Omar; Curran, Patrick; Richards, Matthew; Saradjian, Peter; Miller, J Richard; Knemeyer, Ian; Otte, Karin M; Vincent, Stella; Sciammetta, Nunzio; Pasternak, Alexander; Bennett, David Jonathan; Han, Yongxin

Discovery of Potent and Orally Available Bicyclo[1.1.1]pentane-Derived Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitors

发现高效且口服有效的双环[1.1.1]戊烷衍生的吲哚胺-2,3-双加氧酶1 (IDO1) 抑制剂

Pu, Qinglin; Zhang, Hongjun; Guo, Liangqin; Cheng, Mangeng; Doty, Amy C; Ferguson, Heidi; Fradera, Xavier; Lesburg, Charles A; McGowan, Meredeth A; Miller, J Richard; Geda, Prasanthi; Song, Xuelei; Otte, Karin; Sciammetta, Nunzio; Solban, Nicolas; Yu, Wensheng; Sloman, David L; Zhou, Hua; Lammens, Alfred; Neumann, Lars; Bennett, David Jonathan; Pasternak, Alexander; Han, Yongxin

Epitope interactions of monoclonal antibodies targeting CD20 and their relationship to functional properties

靶向CD20的单克隆抗体的表位相互作用及其与功能特性的关系

Klein, Christian; Lammens, Alfred; Schäfer, Wolfgang; Georges, Guy; Schwaiger, Manfred; Mössner, Ekkehard; Hopfner, Karl-Peter; Umaña, Pablo; Niederfellner, Gerhard