日期 影响因子
日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:
–

Appendage- and Scaffold-Diverse Electrophilic and Photoreactive Probes for Integrated Phenotypic Screening-Target Identification Campaigns via a Minimalist Bifunctional Isocyanide

利用极简双功能异氰化物构建具有多样化附属结构和骨架的亲电和光反应探针，用于整合表型筛选-靶标鉴定活动

期刊:ACS Omega
影响因子:4.3
doi:10.1021/acsomega.4c06879
Jackson, Paul A; Kisty, Eleni; Pradhan, Vandan; Swank, Christopher; Bohrer, Luke; Nolan, Tammy L; Weerapana, Eranthie; Lapinsky, David J
发表日期：2024
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Structural studies of the human α(1) glycine receptor via site-specific chemical cross-linking coupled with mass spectrometry.

利用位点特异性化学交联结合质谱法对人类α(1)甘氨酸受体进行结构研究

期刊:Biophysical Reports
影响因子:2.7
doi:10.1016/j.bpr.2024.100184
Veeramachaneni Rathna J, Donelan Chelsee A, Tomcho Kayce A, Aggarwal Shaili, Lapinsky David J, Cascio Michael
Human
发表日期：2024
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Clickable photoaffinity ligands for the human serotonin transporter based on the selective serotonin reuptake inhibitor (S)-citalopram

基于选择性血清素再摄取抑制剂(S)-西酞普兰的用于人类血清素转运蛋白的可点击光亲和配体

期刊:Bioorganic & Medicinal Chemistry Letters
影响因子:2.2
doi:10.1016/j.bmcl.2018.09.029
Yarravarapu, Nageswari; Geffert, Laura; Surratt, Christopher K; Cascio, Michael; Lapinsky, David J
发表日期：2018
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Clickable Photoaffinity Ligands for Metabotropic Glutamate Receptor 5 Based on Select Acetylenic Negative Allosteric Modulators

基于特定乙炔负变构调节剂的代谢型谷氨酸受体5可点击光亲和配体

期刊:ACS Chemical Biology
影响因子:3.8
doi:10.1021/acschembio.6b00026
Gregory, Karen J; Velagaleti, Ranganadh; Thal, David M; Brady, Ryan M; Christopoulos, Arthur; Conn, P Jeffrey; Lapinsky, David J
信号转导
代谢
发表日期：2016
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Novel Azido-Iodo Photoaffinity Ligands for the Human Serotonin Transporter Based on the Selective Serotonin Reuptake Inhibitor (S)-Citalopram

基于选择性血清素再摄取抑制剂（S）-西酞普兰的新型叠氮-碘光亲和配体用于人类血清素转运蛋白

期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.5b00682
Kumar, Vivek; Yarravarapu, Nageswari; Lapinsky, David J; Perley, Danielle; Felts, Bruce; Tomlinson, Michael J; Vaughan, Roxanne A; Henry, L Keith; Lever, John R; Newman, Amy Hauck
Human
发表日期：2015
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(±)-2-(N-tert-Butylamino)-3'-[(125)I]-iodo-4'-azidopropiophenone: a dopamine transporter and nicotinic acetylcholine receptor photoaffinity ligand based on bupropion (Wellbutrin, Zyban)

(±)-2-(N-叔丁基氨基)-3'-[(125)I]-碘-4'-叠氮丙苯酮：一种基于安非他酮（Wellbutrin，Zyban）的多巴胺转运体和尼古丁乙酰胆碱受体光亲和配体

期刊:Bioorganic & Medicinal Chemistry Letters
影响因子:2.2
doi:10.1016/j.bmcl.2011.10.086
Lapinsky, David J; Aggarwal, Shaili; Nolan, Tammy L; Surratt, Christopher K; Lever, John R; Acharya, Rejwi; Vaughan, Roxanne A; Pandhare, Akash; Blanton, Michael P
信号转导
发表日期：2012
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