日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Radioiodination of Two Carborane-Based Dual Cyclooxygenase-2/5-Lipoxygenase Inhibitors and Their In Vitro and In Vivo Evaluation

两种基于碳硼烷的双重环氧合酶-2/5-脂氧合酶抑制剂的放射性碘化及其体外和体内评价

Schädlich, Jonas; Ullrich, Martin; Haase-Kohn, Cathleen; Wodtke, Robert; Braun, Sebastian; Molitor, Maximilian; Hofmann, Bettina; Steinhilber, Dieter; Kopka, Klaus; Hey-Hawkins, Evamarie; Pietzsch, Jens; Laube, Markus

Deciphering the Tumor Uptake of Heterobivalent (SST(2)/Albumin) [(64)Cu]Cu-NODAGA-cLAB-TATEs

解析异二价 (SST(2)/白蛋白) [(64)Cu]Cu-NODAGA-cLAB-TATEs 的肿瘤摄取

Brandt, Florian; Ullrich, Martin; Laube, Markus; Löser, Reik; Kotzerke, Jörg; Kopka, Klaus; Pietzsch, Jens; van den Hoff, Jörg; Wodtke, Robert

PET and SPECT Tracer Development via Copper-Mediated Radiohalogenation of Divergent and Stable Aryl-Boronic Esters

利用铜介导的放射性卤化反应开发不同类型和稳定的芳基硼酸酯的PET和SPECT示踪剂

Craig, Austin; Sachse, Frederik J; Laube, Markus; Brandt, Florian; Kopka, Klaus; Stadlbauer, Sven

Exploring a Nitric Oxide-Releasing Celecoxib Derivative as a Potential Modulator of Bone Healing: Insights from Ex Vivo and In Vivo Imaging Experiments

探索一氧化氮释放型塞来昔布衍生物作为骨愈合潜在调节剂的作用:来自离体和体内成像实验的启示

Neuber, Christin; Niedenzu, Luisa; Schulze, Sabine; Laube, Markus; Hofheinz, Frank; Rammelt, Stefan; Pietzsch, Jens

Exploring the Role of Peripheral Macrophages in Glioma Progression: The Metabolic Significance of Cyclooxygenase-2 (COX-2).

探索外周巨噬细胞在胶质瘤进展中的作用:环氧合酶-2 (COX-2) 的代谢意义

Pietzsch Jens, Toussaint Magali, Donat Cornelius Kurt, Doctor Alina, Meister Sebastian, Wodtke Johanna, Laube Markus, Hofheinz Frank, Rix Jan, Deuther-Conrad Winnie, Haase-Kohn Cathleen

In Vitro Characterization of the Published Glypican-3-Targeting Peptide TJ12P2 Reveals a Lack of Specificity and Potency.

已发表的 Glypican-3 靶向肽 TJ12P2 的体外表征显示其缺乏特异性和效力。

Burger Eva-Maria, Hill Charlice, Wodtke Robert, Zarschler Kristof, Laube Markus, Donat Cornelius K, Hauser Sandra, Kopka Klaus, Pietzsch Jens, Stadlbauer Sven

Novel Ruthenacarborane-NSAID Conjugates

新型钌碳硼烷-非甾体抗炎药缀合物

Sonam, Sonam; Mojić, Marija; Gordić, Vuk; Laube, Markus; Schädlich, Jonas; Pietzsch, Jens; Nicoara, Adrian; Gaina, Luiza; Mijatović, Sanja; Maksimović-Ivanić, Danijela; Kaluđerović, Goran N; Hey-Hawkins, Evamarie

Carborane-Based Analogs of Celecoxib and Flurbiprofen, their COX Inhibition Potential, and COX Selectivity Index

基于碳硼烷的塞来昔布和氟比洛芬类似物、其COX抑制潜力和COX选择性指数

Ueberham, Lea; Schädlich, Jonas; Schramke, Kim; Braun, Sebastian; Selg, Christoph; Laube, Markus; Lönnecke, Peter; Pietzsch, Jens; Hey-Hawkins, Evamarie

Carborane Conjugates with Ibuprofen, Fenoprofen and Flurbiprofen: Synthesis, Characterization, COX Inhibition Potential and In Vitro Activity.

布洛芬、非诺洛芬和氟比洛芬的碳硼烷缀合物:合成、表征、COX抑制潜力和体外活性

Sonam Sonam, Jelača Sanja, Laube Markus, Schädlich Jonas, Pietzsch Jens, Maksimović-Ivanić Danijela, Mijatović Sanja, Kaluđerović Goran N, Hey-Hawkins Evamarie

Advances in Diclofenac Derivatives: Exploring Carborane-Substituted N-Methyl and Nitrile Analogs for Anticancer Therapy.

双氯芬酸衍生物的研究进展:探索碳硼烷取代的N-甲基和腈类似物在抗癌治疗中的应用

Selg Christoph, Schuster Robert, Kazimir Aleksandr, Lönnecke Peter, Wolniewicz Mara, Schädlich Jonas, Laube Markus, Pietzsch Jens, Gordić Vuk, Krajnović Tamara, Mijatović Sanja, Maksimović-Ivanić Danijela, Hey-Hawkins Evamarie