日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Crystal structures of the selenoprotein glutathione peroxidase 4 in its apo form and in complex with the covalently bound inhibitor ML162

硒蛋白谷胱甘肽过氧化物酶 4 的载脂蛋白形式及其与共价结合抑制剂 ML162 的复合物的晶体结构

Dieter Moosmayer, André Hilpmann, Jutta Hoffmann, Lennart Schnirch, Katja Zimmermann, Volker Badock, Laura Furst, John K Eaton, Vasanthi S Viswanathan, Stuart L Schreiber, Stefan Gradl, Roman C Hillig

Selective covalent targeting of GPX4 using masked nitrile-oxide electrophiles

使用掩蔽的腈氧化物亲电试剂对 GPX4 进行选择性共价靶向

John K Eaton, Laura Furst, Richard A Ruberto, Dieter Moosmayer, André Hilpmann, Matthew J Ryan, Katja Zimmermann, Luke L Cai, Michael Niehues, Volker Badock, Anneke Kramm, Sixun Chen, Roman C Hillig, Paul A Clemons, Stefan Gradl, Claire Montagnon, Kiel E Lazarski, Sven Christian, Besnik Bajrami, Rol

Genomic Activation of PPARG Reveals a Candidate Therapeutic Axis in Bladder Cancer

PPARG 的基因组激活揭示了膀胱癌的候选治疗轴

Jonathan T Goldstein, Ashton C Berger, Juliann Shih, Fujiko F Duke, Laura Furst, David J Kwiatkowski, Andrew D Cherniack, Matthew Meyerson, Craig A Strathdee