日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A mammalian, glutaminase-free asparaginase enhances venetoclax activity in preclinical AML models with chromosome 7 deletion

一种不含谷氨酰胺酶的哺乳动物天冬酰胺酶可增强维奈托克在染色体 7 缺失的临床前 AML 模型中的活性

Majid, Dhabya; Wang, Zhe; Schalk, Amanda M; Yuan, Bin; Tatarata, Qi Zhang; Root, Jessica L; Garza, Araceli Isabella; Yassouf, Mhd Yousuf; Gamal, Basant T; Feri-Borgogno, Sammy; Nguyen, Annie Hoai; Konopleva, Marina; Peeters, Evelien; Su, Ying; Reville, Patrick K; Ravandi-Kashani, Farhad; Lavie, Arnon; Abbas, Hussein A

A human-like glutaminase-free asparaginase is highly efficacious in ASNS(low) leukemia and solid cancer mouse xenograft models.

人类样无谷氨酰胺酶的天冬酰胺酶在 ASNS(low) 白血病和实体癌小鼠异种移植模型中具有很高的疗效

Van Trimpont Maaike, Schalk Amanda M, Hofkens Kenneth, Peeters Evelien, T'Sas Sara, Vandemeulebroecke Katrien, Su Ying, De Loera Ashley, Garcia Alyssa, Chen Hui, Lammens Tim, Van Vlierberghe Pieter, Goossens Steven, Lavie Arnon

In vivo stabilization of a less toxic asparaginase variant leads to a durable antitumor response in acute leukemia

体内稳定毒性较低的天冬酰胺酶变体可导致急性白血病产生持久的抗肿瘤反应。

Van Trimpont, Maaike; Schalk, Amanda M; De Visser, Yanti; Nguyen, Hien Anh; Reunes, Lindy; Vandemeulebroecke, Katrien; Peeters, Evelien; Su, Ying; Lee, Hyun; Lorenzi, Philip L; Chan, Wai-Kin; Mondelaers, Veerle; De Moerloose, Barbara; Lammens, Tim; Goossens, Steven; Van Vlierberghe, Pieter; Lavie, Arnon

The spleen as a sanctuary site for residual leukemic cells following ABT-199 monotherapy in ETP-ALL

在ETP-ALL中,ABT-199单药治疗后,脾脏成为残留白血病细胞的庇护所。

Di Grande, Alessandra; Peirs, Sofie; Donovan, Paul D; Van Trimpont, Maaike; Morscio, Julie; Lintermans, Beatrice; Reunes, Lindy; Vandamme, Niels; Goossens, Steven; Nguyen, Hien Anh; Lavie, Arnon; Lock, Richard B; Prehn, Jochen H M; Van Vlierberghe, Pieter; Ní Chonghaile, Triona

pH-Dependent Mechanisms of Influenza Infection Mediated by Hemagglutinin

血凝素介导的流感病毒感染的pH依赖性机制

Caffrey, Michael; Lavie, Arnon

Metabolic Modifier Screen Reveals Secondary Targets of Protein Kinase Inhibitors within Nucleotide Metabolism

代谢调节剂筛选揭示核苷酸代谢中蛋白激酶抑制剂的次要靶点

Abt, Evan R; Rosser, Ethan W; Durst, Matthew A; Lok, Vincent; Poddar, Soumya; Le, Thuc M; Cho, Arthur; Kim, Woosuk; Wei, Liu; Song, Janet; Capri, Joseph R; Xu, Shili; Wu, Nanping; Slavik, Roger; Jung, Michael E; Damoiseaux, Robert; Czernin, Johannes; Donahue, Timothy R; Lavie, Arnon; Radu, Caius G

Structure of avian influenza hemagglutinin in complex with a small molecule entry inhibitor

禽流感血凝素与小分子入侵抑制剂复合物的结构

Antanasijevic, Aleksandar; Durst, Matthew A; Cheng, Han; Gaisina, Irina N; Perez, Jasmine T; Manicassamy, Balaji; Rong, Lijun; Lavie, Arnon; Caffrey, Michael

Identification of a pH sensor in Influenza hemagglutinin using X-ray crystallography

利用X射线晶体衍射法鉴定流感病毒血凝素中的pH传感器

Antanasijevic, Aleksandar; Durst, Matthew A; Lavie, Arnon; Caffrey, Michael

Probing the metastable state of influenza hemagglutinin

探究流感血凝素的亚稳态

Kingsley, Carolyn N; Antanasijevic, Aleksandar; Palka-Hamblin, Helena; Durst, Matthew; Ramirez, Benjamin; Lavie, Arnon; Caffrey, Michael

Discovery of human-like L-asparaginases with potential clinical use by directed evolution.

通过定向进化发现具有潜在临床应用价值的类人L-天冬酰胺酶

Rigouin Coraline, Nguyen Hien Anh, Schalk Amanda M, Lavie Arnon