日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

N-Branched Tricyclic Guanidines as Novel Melanocortin-3 Receptor Agonists and Melanocortin-4 Receptor Antagonists

N-支链三环胍类化合物作为新型黑皮质素-3受体激动剂和黑皮质素-4受体拮抗剂

Weirath, Nicholas A; Zajac, Jonathan W P; Donow, Haley M; Lavoi, Travis M; Pinilla, Clemencia; Santos, Radleigh G; Prajapati, Ritu; Speth, Robert; Ericson, Mark D; Sarupria, Sapna; Giulianotti, Marcello A; Haskell-Luevano, Carrie

Structure-Activity Relationship of Pyrrolidine Pentamine Derivatives as Inhibitors of the Aminoglycoside 6'- N-Acetyltransferase Type Ib

吡咯烷五胺衍生物作为氨基糖苷类 6'-N-乙酰转移酶 Ib 型抑制剂的构效关系

Jan Sklenicka, Tung Tran, Maria S Ramirez, Haley M Donow, Angel J Magaña, Travis LaVoi, Yasir Mamun, Verónica Jimenez, Prem Chapagain, Radleigh Santos, Clemencia Pinilla, Marc A Giulianotti, Marcelo E Tolmasky

The co-creation, initial piloting, and protocol for a cluster randomised controlled trial of a coach-led positive body image intervention for girls in sport

共同创建、初步试点和制定一项针对运动中女孩的由教练主导的积极身体形象干预的整群随机对照试验方案

Matheson, E L; Schneider, J; Tinoco, A; Gentili, C; Silva-Breen, H; LaVoi, N M; White, P; Diedrichs, P C

The Parallel Structure-Activity Relationship Screening of Three Compounds Identifies the Common Agonist Pharmacophore of Pyrrolidine Bis-Cyclic Guanidine Melanocortin-3 Receptor (MC3R) Small-Molecule Ligands

三种化合物的平行构效关系筛选鉴定出吡咯烷双环胍类黑皮质素-3受体(MC3R)小分子配体的共同激动剂药效团

Mark D Ericson, Katie T Freeman, Travis M LaVoi, Haley M Donow, Radleigh G Santos, Marc A Giulianotti, Clemencia Pinilla, Richard A Houghten, Carrie Haskell-Luevano

Functional Mixture-Based Positional Scan Identifies a Library of Antagonist Tetrapeptide Sequences (LAtTeS) with Nanomolar Potency for the Melanocortin-4 Receptor and Equipotent with the Endogenous AGRP(86-132) Antagonist

基于功能混合物的定位扫描可识别出具有纳摩尔级黑皮质素-4 受体效力并与内源性 AGRP(86-132) 拮抗剂等效效力的拮抗剂四肽序列 (LAtTeS) 库

Mark D Ericson, Skye R Doering, Courtney M Larson, Katie T Freeman, Travis M LaVoi, Haley M Donow, Radleigh G Santos, Rachel H Cho, Zoe M Koerperich, Marc A Giulianotti, Clemencia Pinilla, Richard A Houghten, Carrie Haskell-Luevano

Discovery of Nanomolar Melanocortin-3 Receptor (MC3R)-Selective Small Molecule Pyrrolidine Bis-Cyclic Guanidine Agonist Compounds Via a High-Throughput "Unbiased" Screening Campaign

通过高通量“无偏”筛选活动发现纳摩尔级黑素皮质素-3受体(MC3R)选择性小分子吡咯烷双环胍激动剂化合物

Doering, Skye R; Freeman, Katie; Debevec, Ginamarie; Geer, Phaedra; Santos, Radleigh G; Lavoi, Travis M; Giulianotti, Marc A; Pinilla, Clemencia; Appel, Jon R; Houghten, Richard A; Ericson, Mark D; Haskell-Luevano, Carrie

Inhibition of Aminoglycoside 6'- N-acetyltransferase Type Ib (AAC(6')-Ib): Structure-Activity Relationship of Substituted Pyrrolidine Pentamine Derivatives as Inhibitors

氨基糖苷类 6'- N-乙酰转移酶 Ib 型 (AAC(6')-Ib) 的抑制:取代吡咯烷五胺衍生物作为抑制剂的构效关系

Kenneth Rocha, Jesus Magallon, Craig Reeves, Kimberly Phan, Peter Vu, Crista L Oakley-Havens, Stella Kwan, Maria Soledad Ramirez, Travis LaVoi, Haley Donow, Prem Chapagain, Radleigh Santos, Clemencia Pinilla, Marc A Giulianotti, Marcelo E Tolmasky

Re-thinking Women's Sport Research: Looking in the Mirror and Reflecting Forward

重新思考女子体育研究:反思与展望

Lebel, Katie; Mumcu, Ceyda; Pegoraro, Ann; LaVoi, Nicole M; Lough, Nancy; Antunovic, Dunja

A Novel Probe for Spliceosomal Proteins that Induces Autophagy and Death of Melanoma Cells Reveals New Targets for Melanoma Drug Discovery

诱导黑色素瘤细胞自噬和死亡的剪接体蛋白新型探针揭示了黑色素瘤药物研发的新靶点

Manikandan Palrasu, Anna M Knapinska, Juan Diez, Lyndsay Smith, Travis LaVoi, Marc Giulianotti, Richard A Houghten, Gregg B Fields, Dmitriy Minond

Direct Phenotypic Screening in Mice: Identification of Individual, Novel Antinociceptive Compounds from a Library of 734,821 Pyrrolidine Bis-piperazines

小鼠直接表型筛选:从包含 734,821 个吡咯烷双哌嗪的化合物库中鉴定出单个新型镇痛化合物

Houghten, Richard A; Ganno, Michelle L; McLaughlin, Jay P; Dooley, Colette T; Eans, Shainnel O; Santos, Radleigh G; LaVoi, Travis; Nefzi, Adel; Welmaker, Greg; Giulianotti, Marc A; Toll, Lawrence