日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

1'-Cyanocytidine-5'-isobutyryl is a potent SARS-CoV-2 inhibitor in culture and infected Syrian hamsters

1'-氰胞苷-5'-异丁酰基在体外培养和感染叙利亚仓鼠中均表现出对SARS-CoV-2的强效抑制作用。

Amblard, Franck; Kasthuri, Mahesh; LeCher, Julia C; Tao, Sijia; De, Ramyani; Abdelnabi, Rana; Marko, Ingrid; Zhou, Longhu; Li, Chengwei; Shi, Junxing; Goh, Shu Ling; Downs-Bowen, Jessica; Bassit, Leda; Hurwitz, Selwyn; Zandi, Keivan; McBrayer, Tamara; Weynand, Birgit; Johnson, Kenneth A; Neyts, Johan; Schinazi, Raymond F

Combating yellow fever virus with 7-deaza-7-fluoro-2'-C-methyladenosine

用7-脱氮-7-氟-2'-C-甲基腺苷对抗黄热病毒

LeCher, Julia C; Costa, Vivian Vasconcelos; Rust, Lauren N; Bassit, Leda C; Patel, Dharmeshkumar; Rezaei, Sahar; Moua, Justin; Santos, Felipe Rocha da Silva; Goncalves, Matheus Rodrigues; Queroz-Junior, Celso Martins; Marim, Fernanda Martins; Zhou, Longhu; Lee, Sujin; McBrayer, Tamara; De, Ramyani; Azadi, Niloufar; Salman, Mohammad; Zandi, Keivan; Amblard, Franck; Burwitz, Benjamin; Teixeira, Mauro M; Schinazi, Raymond F

Synthesis and biological evaluation of novel peptidomimetic inhibitors of the coronavirus 3C-like protease.

冠状病毒3C样蛋白酶新型肽模拟抑制剂的合成及生物学评价

Amblard Franck, LeCher Julia C, De Ramyani, Zhou Shaoman, Liu Peng, Goh Shu Ling, Tao Sijia, Patel Dharmeshkumar, Downs-Bowen Jessica, Zandi Keivan, Zhang Huanchun, Chaudhry Gitika, McBrayer Tamara, Muczynski Michael, Al-Homoudi Abdullah, Engel Joseph, Lan Shuiyun, Sarafianos Stefan G, Kovari Ladislau C, Schinazi Raymond F

Synthesis of 4'-Substituted Carbocyclic Uracil Derivatives and Their Monophosphate Prodrugs as Potential Antiviral Agents

4'-取代碳环尿嘧啶衍生物及其单磷酸前药的合成及其作为潜在抗病毒药物的研究

Biteau, Nicolas G; Amichai, Sarah A; Azadi, Niloufar; De, Ramyani; Downs-Bowen, Jessica; Lecher, Julia C; MacBrayer, Tamara; Schinazi, Raymond F; Amblard, Franck

Utilization of a cell-penetrating peptide-adaptor for delivery of human papillomavirus protein E2 into cervical cancer cells to arrest cell growth and promote cell death

利用细胞穿透肽-适配器将人乳头瘤病毒蛋白E2递送至宫颈癌细胞,以抑制细胞生长并促进细胞死亡

LeCher, Julia C; Didier, Hope L; Dickson, Robert L; Slaughter, Lauren R; Bejarano, Juana C; Ho, Steven; Nowak, Scott J; Chrestensen, Carol A; McMurry, Jonathan L

Discovery of a 2'-Fluoro,2'-Bromouridine Phosphoramidate Prodrug Exhibiting Anti-Yellow Fever Virus Activity in Culture and in Mice

发现一种2'-氟-2'-溴尿苷磷酰胺前药在体外培养和小鼠体内均表现出抗黄热病毒活性

LeCher, Julia C; Zandi, Keivan; Costa, Vivian Vasconcelos; Amblard, Franck; Tao, Sijia; Patel, Dharmeshkumar; Lee, Sujin; da Silva Santos, Felipe Rocha; Goncalves, Matheus Rodrigues; Queroz-Junior, Celso Martins; Marim, Fernanda Martins; Musall, Katie; Goh, Shu Ling; McBrayer, Tamara; Downs-Bowen, Jessica; De, Ramyani; Azadi, Niloufar; Kohler, James; Teixeira, Mauro Martins; Schinazi, Raymond F

Breaking in and busting out: cell-penetrating peptides and the endosomal escape problem

突破与逃脱:细胞穿透肽与内体逃逸问题

LeCher, Julia C; Nowak, Scott J; McMurry, Jonathan L