日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Biological and Structural Analyses of New Potent Allosteric Inhibitors of HIV-1 Integrase

HIV-1 整合酶新型强效变构抑制剂的生物学和结构分析

Damien Bonnard #, Erwann Le Rouzic #, Matthew R Singer #, Zhe Yu, Frédéric Le Strat, Claire Batisse, Julien Batisse, Céline Amadori, Sophie Chasset, Valerie E Pye, Stéphane Emiliani, Benoit Ledoussal, Marc Ruff, François Moreau, Peter Cherepanov, Richard Benarous

Structure-function analyses unravel distinct effects of allosteric inhibitors of HIV-1 integrase on viral maturation and integration

结构-功能分析揭示了HIV-1整合酶变构抑制剂对病毒成熟和整合的不同影响

Bonnard, Damien; Le Rouzic, Erwann; Eiler, Sylvia; Amadori, Céline; Orlov, Igor; Bruneau, Jean-Michel; Brias, Julie; Barbion, Julien; Chevreuil, Francis; Spehner, Danièle; Chasset, Sophie; Ledoussal, Benoit; Moreau, François; Saïb, Ali; Klaholz, Bruno P; Emiliani, Stéphane; Ruff, Marc; Zamborlini, Alessia; Benarous, Richard

The HIV-1 integrase-LEDGF allosteric inhibitor MUT-A: resistance profile, impairment of virus maturation and infectivity but without influence on RNA packaging or virus immunoreactivity

HIV-1整合酶-LEDGF变构抑制剂MUT-A:耐药性特征,损害病毒成熟和感染性,但不影响RNA包装或病毒免疫反应性

Amadori, Céline; van der Velden, Yme Ubeles; Bonnard, Damien; Orlov, Igor; van Bel, Nikki; Le Rouzic, Erwann; Miralles, Laia; Brias, Julie; Chevreuil, Francis; Spehner, Daniele; Chasset, Sophie; Ledoussal, Benoit; Mayr, Luzia; Moreau, François; García, Felipe; Gatell, José; Zamborlini, Alessia; Emiliani, Stéphane; Ruff, Marc; Klaholz, Bruno P; Moog, Christiane; Berkhout, Ben; Plana, Montserrat; Benarous, Richard

Downregulation of renal AQP2 water channel and NKCC2 in mice lacking the apical Na+-H+ exchanger NHE3

缺乏顶端Na+-H+交换器NHE3的小鼠肾脏AQP2水通道和NKCC2表达下调

Amlal, Hassane; Ledoussal, Clara; Sheriff, Sulaiman; Shull, Gary E; Soleimani, Manoocher