Optimization of Indole- and Pyrazole-fused Glycyrrhetinic Acid Derivatives as Potent PTP1B Inhibitors: In Silico, In Vitro, In Vivo, and Metabolomic Studies
吲哚和吡唑稠合甘草次酸衍生物作为强效PTP1B抑制剂的优化:计算机模拟、体外、体内和代谢组学研究
期刊:ACS Bio & Med Chem Au
影响因子:4.3
doi:10.1021/acsbiomedchemau.5c00164
López-Sánchez, Mitzi; Mendoza-Mota, Hannya; De-la-Cruz-Martínez, Ledy; Matadamas-Martínez, Félix; Torres-Chacón, Diana Laura; Martínez-Arellano, Rosendo; Palacios-Espinosa, Juan Francisco; Pérez-Villanueva, Jaime; González-Andrade, Martin; Páez-Franco, José Carlos; Almanza-Pérez, Julio César; Cortés-Benítez, Francisco