日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Optimization of Prodiginines as Single-Dose Curative Antimalarials

优化灵菌红素类药物作为单剂量治愈性抗疟药

Kumar, Amrendra; Li, Yuexin; Zhang, Xiaowei; Gaddam, Mahesh; Caridha, Diana; Madejczyk, Michael S; Jin, Xiannu; Dennis, William E; Chetree, Ravi; Blount, Cameron; DeLuca, Jesse; Vuong, Chau; Kudyba, Karl; Roncal, Norma; Ashraf, Kutub; Lee, Patricia J; Pannone, Kristina; Leed, Susan; Dinh, Hieu T; Mdaki, Kennedy; Navarrete, Kimberly; Charlton, Jordan; Binauhan, Angely J; Qahash, Tarrick; Kibe, Kevin Mugambi; Shoue, Douglas A; Checkley, Lisa; Ferdig, Michael T; Chim-Ong, Anongruk; Cui, Liwang; Orena, Stephen; Byaruhanga, Oswald; Assimwe, Jackson; Tibagambirwa, Innocent; Chithanna, Sivanna; Dodean, Rozalia A; Legac, Jennifer; Kreutzfeld, Oriana; Rosenthal, Philip J; Cooper, Roland A; Reynolds, Kevin A; Roth, Alison; Kelly, Jane X; Kancharla, Papireddy

Maintaining capital discipline in the rush to net-zero energy systems

在迈向净零能源系统的浪潮中保持资本纪律

Greig, Chris; Techau, Michala; Leed, Andreas; Budzier, Alexander

Acridone Prodrugs with Enhanced Dual-Stage Antimalarial Efficacy

具有增强双阶段抗疟功效的吖啶酮前药

Dodean, Rozalia A; Li, Yuexin; Zhang, Xiaowei; Kumar, Amrendra; Pou, Sovitj; W Winter, Rolf; Liebman, Katherine M; Zakharov, Lev N; Caridha, Diana; Madejczyk, Michael S; Vuong, Chau; DeLuca, Jesse; Chin, Geoffrey; Kudyba, Karl; McEnearney, Sharon; Jin, Xiannu; Dennis, William E; Chetree, Ravi; Blount, Cameron; Pannone, Kristina; Dinh, Hieu T; Mdaki, Kennedy; Leed, Susan; Lee, Patricia J; Roth, Alison; Kancharla, Papireddy; Kelly, Jane X

Identification of Substituted 4-Aminocinnolines as Broad-Spectrum Antiparasitic Agents

鉴定取代的4-氨基喹啉类化合物作为广谱抗寄生虫药物

Spaulding, Andrew; Sharma, Amrita; Giardini, Miriam A; Hoffman, Benjamin; Bernatchez, Jean A; McCall, Laura-Isobel; Calvet, Claudia M; Ackermann, Jasmin; Souza, Julia M; Thomas, Diane; Millard, Caroline C; Devine, William G; Singh, Baljinder; Silva, Everton M; Leed, Susan E; Roncal, Norma E; Penn, Erica C; Erath, Jessey; Kumar, Gaurav; Sepulveda, Yadira; Garcia, Arnold; Rodriguez, Ana; El-Sakkary, Nelly; Sciotti, Richard J; Campbell, Robert F; Momper, Jeremiah D; McKerrow, James H; Caffrey, Conor R; Siqueira-Neto, Jair L; Pollastri, Michael P; Mensa-Wilmot, Kojo; Ferrins, Lori

In vitro activity and in vivo efficacy of omadacycline against Plasmodium species.

奥马环素对疟原虫的体外活性和体内疗效

Madejczyk Michael S, Leed Susan E, Kudyba Karl, Roth Alison, Martin Monica L, Lee Patricia, Anastasiou Diane, Pierce Jessica V, Serio Alisa W, Caridha Diana

Potent Acridone Antimalarial against All Three Life Stages of Plasmodium

强效抗疟药吖啶酮,可对抗疟原虫所有三个生命阶段

Kancharla, Papireddy; Dodean, Rozalia A; Li, Yuexin; Zhang, Xiaowei; Kelly, Sean; Charlton, Jordan; Binauhan, Angley; Garcia, Laurize; Caridha, Diana; Madejczyk, Michael S; Jin, Xiannu; Dennis, William E; Kudyba, Karl; McEnearney, Sharon; Lee, Partricia J; Blount, Cameron; DeLuca, Jesse; Vuong, Chua; Pannone, Kristina; Dinh, Hieu T; Mdaki, Kennedy; Leed, Susan; Martin, Monica L; Pybus, Brandon S; Chimong, Anongruk; Cui, Liwang; Vega-Rodriguez, Joel; Okitwi, Martin; Kreutzfeld, Oriana; Docan, Christina; Green, Carol; Liu, Ying; Agulay, Aaron; Mirsalis, Jon; Farrell, Sarah N; McFadden, Geoffrey I; Goodman, Christopher D; Probst, Alexandra S; Nilsen, Aaron; Catteruccia, Flaminia; Rosenthal, Philip J; Riscoe, Michael; Cooper, Roland; Roth, Alison; Kelly, Jane

Targeting NEDD9-SH3 with a Covalent Peptide Controls Endothelial Phenotype.

利用共价肽靶向NEDD9-SH3可控制内皮细胞表型

Samokhin Andriy O, Seo Hyuk-Soo, Leed Alison, Hajian Behnoush, Bird Gregory H, McKinney David C, Saha Progyaparamita, Daum Jacqueline, Moroco Jamie A, Yehl Jenna, Kornfilt David, Szczeniowski Anna, Petrunak Elyse, Horner Steven, Kalin Jay H, Leymarie Nancy, Kaushik Virendar K, Walensky Loren D, Cole Philip A, Oldham William M, Steinhauser Matthew L, Dhe-Paganon Sirano, Maron Bradley A

Phenotypic screening converges on CDK9 inhibition as a therapeutic strategy in translocation renal cell carcinoma.

表型筛选结果表明,CDK9 抑制是易位性肾细胞癌的一种治疗策略

Thapa Dharma R, Deodhar Riva, Skepner Adam, Konda Prathyusha, Zhou Meng, Bluck Joseph, Pichlo Christian, Cui Yantong, Stocker Paige, Khanna Prateek, Li Jiao, Tsai Jonathan M, Leed Alison, Gould Sandy, Alimova Maria, Friedrich Dhana, Cheah Jaime H, Rupaimoole Rajesha, Guicherit Oivin, Viswanathan Srinivas R

Novel hydrazone compounds with broad-spectrum antiplasmodial activity and synergistic interactions with antimalarial drugs

具有广谱抗疟原虫活性并与抗疟药物有协同作用的新型腙化合物

Angélica M Rosado-Quiñones, Emilee E Colón-Lorenzo, Zarna Rajeshkumar Pala, Jürgen Bosch, Karl Kudyba, Heather Kudyba, Susan E Leed, Norma Roncal, Abel Baerga-Ortiz, Abiel Roche-Lima, Yamil Gerena, David A Fidock, Alison Roth, Joel Vega-Rodríguez #, Adelfa E Serrano #

DDDR-05. SPATIALLY RESOLVED DRUG SENSITIVITY PROFILING IN GLIOBLASTOMA

DDDR-05. 胶质母细胞瘤的空间分辨药物敏感性分析

Kumar, Amrendra; Li, Yuexin; Dodean, Rozalia A; Roth, Alison; Caridha, Diana; Madejczyk, Michael S; Jin, Xiannu; Dennis, William E; Lee, Patricia J; Pybus, Brandon S; Martin, Monica; Pannone, Kristina; Dinh, Hieu T; Blount, Cameron; Chetree, Ravi; DeLuca, Jesse; Evans, Martin; Nadeau, Robert; Vuong, Chau; Leed, Susan; Black, Chad; Sousa, Jason; Nolan, Christina; Ceja, Frida G; Rasmussen, Stephanie A; Tumwebaze, Patrick K; Rosenthal, Philip J; Cooper, Roland A; Rottmann, Matthias; Orjuela-Sanchez, Pamela; Meister, Stephan; Winzeler, Elizabeth A; Delves, Michael J; Matthews, Holly; Baum, Jake; Kirby, Robert W; Burrows, Jeremy N; Duffy, James; Peyton, David H; Reynolds, Kevin A; Kelly, Jane X; Kancharla, Papireddy; Buck, Alicia; Lee, Sohyon; Wegmann, Rebekka; Mena, Julien; Vasella, Flavio; Friesen, Julia; Regli, Luca; Le Rhun, Emilie; Zeitlberger, Anna Maria; Neidert, Marian Christoph; Tatari, Nazanin; Hutter, Gregor; Weller, Michael; Snijder, Berend; Weiss, Tobias