日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of Substituted 4-Aminocinnolines as Broad-Spectrum Antiparasitic Agents

鉴定取代的4-氨基喹啉类化合物作为广谱抗寄生虫药物

Spaulding, Andrew; Sharma, Amrita; Giardini, Miriam A; Hoffman, Benjamin; Bernatchez, Jean A; McCall, Laura-Isobel; Calvet, Claudia M; Ackermann, Jasmin; Souza, Julia M; Thomas, Diane; Millard, Caroline C; Devine, William G; Singh, Baljinder; Silva, Everton M; Leed, Susan E; Roncal, Norma E; Penn, Erica C; Erath, Jessey; Kumar, Gaurav; Sepulveda, Yadira; Garcia, Arnold; Rodriguez, Ana; El-Sakkary, Nelly; Sciotti, Richard J; Campbell, Robert F; Momper, Jeremiah D; McKerrow, James H; Caffrey, Conor R; Siqueira-Neto, Jair L; Pollastri, Michael P; Mensa-Wilmot, Kojo; Ferrins, Lori

In vitro activity and in vivo efficacy of omadacycline against Plasmodium species.

奥马环素对疟原虫的体外活性和体内疗效

Madejczyk Michael S, Leed Susan E, Kudyba Karl, Roth Alison, Martin Monica L, Lee Patricia, Anastasiou Diane, Pierce Jessica V, Serio Alisa W, Caridha Diana

Anilinoquinoline based inhibitors of trypanosomatid proliferation

基于苯胺喹啉的锥虫增殖抑制剂

Ferrins, Lori; Sharma, Amrita; Thomas, Sarah M; Mehta, Naimee; Erath, Jessey; Tanghe, Scott; Leed, Susan E; Rodriguez, Ana; Mensa-Wilmot, Kojo; Sciotti, Richard J; Gillingwater, Kirsten; Pollastri, Michael P

Assessment of the Worldwide Antimalarial Resistance Network Standardized Procedure for In Vitro Malaria Drug Sensitivity Testing Using SYBR Green Assay for Field Samples with Various Initial Parasitemia Levels

评估全球抗疟疾耐药性网络标准化程序,该程序使用SYBR Green法对具有不同初始寄生虫血症水平的现场样本进行体外疟疾药物敏感性测试

Cheruiyot, Agnes C; Auschwitz, Jennifer M; Lee, Patricia J; Yeda, Redemptah A; Okello, Charles O; Leed, Susan E; Talwar, Mayank; Murthy, Tushar; Gaona, Heather W; Hickman, Mark R; Akala, Hoseah M; Kamau, Edwin; Johnson, Jacob D

EVALUATION OF AROMATIC 6-SUBSTITUTED THIENOPYRIMIDINES AS SCAFFOLDS AGAINST PARASITES THAT CAUSE TRYPANOSOMIASIS, LEISHMANIASIS, AND MALARIA

评价芳香族6-取代噻吩并嘧啶作为抗锥虫病、利什曼病和疟疾寄生虫的骨架化合物

Woodring, Jennifer L; Patel, Gautam; Erath, Jessey; Behera, Ranjan; Lee, Patricia J; Leed, Susan E; Rodriguez, Ana; Sciotti, Richard J; Mensa-Wilmot, Kojo; Pollastri, Michael P

Repurposing human Aurora kinase inhibitors as leads for anti-protozoan drug discovery

将人类Aurora激酶抑制剂重新用于抗原生动物药物研发

Patel, Gautam; Roncal, Norma E; Lee, Patricia J; Leed, Susan E; Erath, Jessey; Rodriguez, Ana; Sciotti, Richard J; Pollastri, Michael P

Design, synthesis, and biological activity of diaryl ether inhibitors of Toxoplasma gondii enoyl reductase

弓形虫烯酰还原酶二芳醚抑制剂的设计、合成及生物活性研究

Cheng, Gang; Muench, Stephen P; Zhou, Ying; Afanador, Gustavo A; Mui, Ernest J; Fomovska, Alina; Lai, Bo Shiun; Prigge, Sean T; Woods, Stuart; Roberts, Craig W; Hickman, Mark R; Lee, Patty J; Leed, Susan E; Auschwitz, Jennifer M; Rice, David W; McLeod, Rima

Development of a triclosan scaffold which allows for adaptations on both the A- and B-ring for transport peptides

开发一种三氯生支架,该支架的A环和B环均可进行改造以适应转运肽。

Muench, Stephen P; Stec, Jozef; Zhou, Ying; Afanador, Gustavo A; McPhillie, Martin J; Hickman, Mark R; Lee, Patty J; Leed, Susan E; Auschwitz, Jennifer M; Prigge, Sean T; Rice, David W; McLeod, Rima

Novel N-benzoyl-2-hydroxybenzamide disrupts unique parasite secretory pathway

新型N-苯甲酰基-2-羟基苯甲酰胺可破坏独特的寄生虫分泌途径

Fomovska, Alina; Huang, Qingqing; El Bissati, Kamal; Mui, Ernest J; Witola, William H; Cheng, Gang; Zhou, Ying; Sommerville, Caroline; Roberts, Craig W; Bettis, Sam; Prigge, Sean T; Afanador, Gustavo A; Hickman, Mark R; Lee, Patty J; Leed, Susan E; Auschwitz, Jennifer M; Pieroni, Marco; Stec, Jozef; Muench, Stephen P; Rice, David W; Kozikowski, Alan P; McLeod, Rima