日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of INCB126503 as a Potent and Selective FGFR2/3 Inhibitor

发现 INCB126503 是一种高效且选择性的 FGFR2/3 抑制剂

Nguyen, Minh H; Wang, Anlai; Truong, Lisa; Zhang, Ke; Ye, Hai-Fen; Zhao, Peng; Horsey, April; Frascella, Michelle; Leffet, Lynn; Federowicz, Kelly; Behshad, Elham; Witten, Michael R; Qi, Chao; Xu, Yao; Jalluri, Ravi; Harris, Jennifer J; Hess, Rodrigo; Sayers, Brian; Lin, Luping; Yeleswaram, Swamy; Zhang, Guofeng; Kim, Sunkyu; Covington, Maryanne; Diamond, Sharon; Yao, Wenqing; Vechorkin, Oleg

Discovery of Orally Bioavailable FGFR2/FGFR3 Dual Inhibitors via Structure-Guided Scaffold Repurposing Approach

通过结构导向的骨架重定位方法发现口服生物利用度高的FGFR2/FGFR3双重抑制剂

Nguyen, Minh H; Ye, Hai-Fen; Xu, Yao; Truong, Lisa; Horsey, April; Zhao, Peng; Styduhar, Evan D; Frascella, Michelle; Leffet, Lynn; Federowicz, Kelly; Behshad, Elham; Wang, Anlai; Zhang, Ke; Witten, Michael R; Qi, Chao; Jalluri, Ravi; Lai, Cheng-Tsung; Atasoylu, Onur; Harris, Jennifer J; Hess, Rodrigo; Lin, Luping; Zhang, Guofeng; Covington, Maryanne; Diamond, Sharon; Yao, Wenqing; Vechorkin, Oleg

INCB24360 (Epacadostat), a Highly Potent and Selective Indoleamine-2,3-dioxygenase 1 (IDO1) Inhibitor for Immuno-oncology

INCB24360(Epacadostat),一种高效且选择性的吲哚胺-2,3-双加氧酶1(IDO1)抑制剂,用于免疫肿瘤学

Yue, Eddy W; Sparks, Richard; Polam, Padmaja; Modi, Dilip; Douty, Brent; Wayland, Brian; Glass, Brian; Takvorian, Amy; Glenn, Joseph; Zhu, Wenyu; Bower, Michael; Liu, Xiangdong; Leffet, Lynn; Wang, Qian; Bowman, Kevin J; Hansbury, Michael J; Wei, Min; Li, Yanlong; Wynn, Richard; Burn, Timothy C; Koblish, Holly K; Fridman, Jordan S; Emm, Tom; Scherle, Peggy A; Metcalf, Brian; Combs, Andrew P

Immunogenicity of H1N1 influenza virus-like particles produced in Nicotiana benthamiana

本氏烟草中产生的H1N1流感病毒样颗粒的免疫原性

Shoji, Yoko; Prokhnevsky, Alex; Leffet, Brett; Vetter, Nancy; Tottey, Stephen; Satinover, Shama; Musiychuk, Konstantin; Shamloul, Moneim; Norikane, Joey; Jones, R Mark; Chichester, Jessica A; Green, Brian J; Streatfield, Stephen J; Yusibov, Vidadi

Potent antisense oligonucleotides to the human multidrug resistance-1 mRNA are rationally selected by mapping RNA-accessible sites with oligonucleotide libraries

利用寡核苷酸文库对RNA可及位点进行定位,可以合理筛选出针对人类多药耐药基因1 mRNA的高效反义寡核苷酸。

Ho, S P; Britton, D H; Stone, B A; Behrens, D L; Leffet, L M; Hobbs, F W; Miller, J A; Trainor, G L