日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Mechanism of beta-arrestin 1 mediated Src activation via Src SH3 domain revealed by cryo-electron microscopy.

冷冻电镜揭示了β-arrestin 1通过Src SH3结构域介导Src激活的机制。

Pakharukova Natalia, Thomas Brittany N, Bansia Harsh, Li Linus, Bassford Dana K, Abzalimov Rinat R, Kim Jihee, Kahsai Alem W, Pani Biswaranjan, Xiao Kunhong, Ochakovski Roni, Liu Shibo, Zhang Xingdong, Ahn Seungkirl, des Georges Amedee, Lefkowitz Robert J

Cardiomyocyte β-arrestins mediate inflammation and cGAS-STING activation in CVB3 viral myocarditis.

心肌细胞β-阻滞蛋白介导CVB3病毒性心肌炎的炎症和cGAS-STING激活。

Lucero Emilio Y, Jiang Haoran, D'Anniballe Vincent, Pakharukova Natalia, Galtes Daniella, Bassford Dana, Jyothidasan Arun, Knowlton Kirk U, Gunn Michael Dee, Lefkowitz Robert J, Rockman Howard A

Small-molecule modulation of β-arrestins

小分子对β-arrestin的调控

Kahsai, Alem W; Pakharukova, Natalia; Kwon, Henry Y; Shah, Kunal S; Liang-Lin, Jason G; Del Real, Caroline T; Shim, Paul J; Lee, Mason A; Ngo, Van A; Shreiber, Bowie N; Liu, Samuel; Schwalb, Allison M; Espinoza, Emmanuel F; Thomas, Brittany N; Kunzle, Cal A; Smith, Jeffrey S; Wang, Jialu; Kim, Jihee; Zhang, Xingdong; Rockman, Howard A; Thomsen, Alex R B; Rein, Lindsay A M; Shi, Lei; Ahn, Seungkirl; Masoudi, Ali; Lefkowitz, Robert J

G Protein-Coupled Receptors: A Century of Research and Discovery

G蛋白偶联受体:一个世纪的研究与发现

Liu, Samuel; Anderson, Preston J; Rajagopal, Sudarshan; Lefkowitz, Robert J; Rockman, Howard A

G protein-coupled receptors: from radioligand binding to cellular signaling

G蛋白偶联受体:从放射性配体结合到细胞信号传导

Rockman, Howard A; Lefkowitz, Robert J

How carvedilol does not activate β(2)-adrenoceptors

卡维地洛如何不激活β(2)-肾上腺素受体

Lefkowitz, Robert J; Rockman, Howard A; Shim, Paul J; Liu, Samuel; Ahn, Seungkirl; Pani, Biswaranjan; Rajagopal, Sudarshan; Shenoy, Sudha K; Bouvier, Michel; Benovic, Jeffrey L; Liggett, Stephen B; Ruffolo, Robert R; Bristow, Michael R; Packer, Milton

Allosteric modulator potentiates β2AR agonist-promoted bronchoprotection in asthma models

变构调节剂增强β2肾上腺素能受体激动剂在哮喘模型中促进的支气管保护作用

Ahn, Seungkirl; Maarsingh, Harm; Walker, Julia Kl; Liu, Samuel; Hegde, Akhil; Sumajit, Hyeje C; Kahsai, Alem W; Lefkowitz, Robert J

Signal transduction at GPCRs: Allosteric activation of the ERK MAPK by β-arrestin

GPCR信号转导:β-arrestin对ERK MAPK的变构激活

Kahsai, Alem W; Shah, Kunal S; Shim, Paul J; Lee, Mason A; Shreiber, Bowie N; Schwalb, Allison M; Zhang, Xingdong; Kwon, Henry Y; Huang, Li-Yin; Soderblom, Erik J; Ahn, Seungkirl; Lefkowitz, Robert J

Loss of biased signaling at a G protein-coupled receptor in overexpressed systems

过表达系统中G蛋白偶联受体偏向性信号的丧失

Li, Angus; Liu, Samuel; Huang, Rennica; Ahn, Seungkirl; Lefkowitz, Robert J

β-Arrestin-Biased Allosteric Modulator Potentiates Carvedilol-Stimulated β Adrenergic Receptor Cardioprotection

β-arrestin偏向性变构调节剂增强卡维地洛刺激的β肾上腺素能受体心脏保护作用

Wang, Jialu; Pani, Biswaranjan; Gokhan, Ilhan; Xiong, Xinyu; Kahsai, Alem W; Jiang, Haoran; Ahn, Seungkirl; Lefkowitz, Robert J; Rockman, Howard A