日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Study of Surface Integrity Evolution During Laser Hardening of 42CrMo4 Steel Using a 4 kW Diode Laser

利用4kW二极管激光器研究42CrMo4钢激光硬化过程中表面完整性的演变

Lazov, Lyubomir; Teirumnieks, Edmunds; Yankov, Emil; Muiznieks, Gatis; Leitans, Armands; Rēvalds, Ritvars; Čapek, Jiří; Trojan, Karel; Prodanov, Prodan; Adijāns, Imants; Kudrjavcevs, Aleksandrs; Sirants, Raimonds

Affinity and Selectivity of Protein-Ligand Recognition: A Minor Chemical Modification Changes Carbonic Anhydrase Binding Profile

蛋白质-配体识别的亲和力和选择性:微小的化学修饰改变碳酸酐酶的结合谱

Zakšauskas, Audrius; Paketurytė-Latvė, Vaida; Janku̅naitė, Alberta; Čapkauskaitė, Edita; Becart, Yann; Smirnov, Alexey; Pospíšilová, Klára; Leitans, Janis; Brynda, Jiří; Kazaks, Andris; Baranauskienė, Lina; Manakova, Elena; Gražulis, Saulius; Kairys, Visvaldas; Tars, Kaspars; Řezáčová, Pavlína; Matulis, Daumantas

Surface Functionalization of ITO for Dual-Mode Hypoxia-Associated Cancer Biomarker Detection.

用于双模式缺氧相关癌症生物标志物检测的ITO表面功能化

Zutis Edmunds, Paidere Gunita, Ruska Rihards, Freimanis Toms, Cipa Janis, Zalubovskis Raivis, Elksne Maira, Tars Kaspars, Kazaks Andris, Leitans Janis, Sarakovskis Anatolijs, Anspoks Andris

Targeted anticancer pre-vinylsulfone covalent inhibitors of carbonic anhydrase IX

靶向抗癌的碳酸酐酶IX前乙烯基砜共价抑制剂

Vaškevičius, Aivaras; Baronas, Denis; Leitans, Janis; Kvietkauskaitė, Agnė; Rukšėnaitė, Audronė; Manakova, Elena; Toleikis, Zigmantas; Kaupinis, Algirdas; Kazaks, Andris; Gedgaudas, Marius; Mickevičiūtė, Aurelija; Juozapaitienė, Vaida; Schiöth, Helgi B; Jaudzems, Kristaps; Valius, Mindaugas; Tars, Kaspars; Gražulis, Saulius; Meyer-Almes, Franz-Josef; Matulienė, Jurgita; Zubrienė, Asta; Dudutienė, Virginija; Matulis, Daumantas

From X-ray crystallographic structure to intrinsic thermodynamics of protein-ligand binding using carbonic anhydrase isozymes as a model system

以碳酸酐酶同工酶为模型体系,研究蛋白质-配体结合的X射线晶体结构及其内在热力学性质

Paketurytė-Latvė, Vaida; Smirnov, Alexey; Manakova, Elena; Baranauskiene, Lina; Petrauskas, Vytautas; Zubrienė, Asta; Matulienė, Jurgita; Dudutienė, Virginija; Čapkauskaitė, Edita; Zakšauskas, Audrius; Leitans, Janis; Gražulis, Saulius; Tars, Kaspars; Matulis, Daumantas

Methyl 2-Halo-4-Substituted-5-Sulfamoyl-Benzoates as High Affinity and Selective Inhibitors of Carbonic Anhydrase IX

2-卤代-4-取代-5-氨磺酰基苯甲酸甲酯作为碳酸酐酶 IX 的高亲和力和选择性抑制剂

Audrius Zakšauskas, Edita Čapkauskaitė, Vaida Paketurytė-Latvė, Alexey Smirnov, Janis Leitans, Andris Kazaks, Elviss Dvinskis, Laimonas Stančaitis, Aurelija Mickevičiūtė, Jelena Jachno, Linas Jezepčikas, Vaida Linkuvienė, Andrius Sakalauskas, Elena Manakova, Saulius Gražulis, Jurgita Matulienė, Kasp

Isoform-Selective Enzyme Inhibitors by Exploring Pocket Size According to the Lock-and-Key Principle

基于锁钥原理,通过探索口袋大小来设计同工酶选择性酶抑制剂

Dudutienė, Virginija; Zubrienė, Asta; Kairys, Visvaldas; Smirnov, Alexey; Smirnovienė, Joana; Leitans, Janis; Kazaks, Andris; Tars, Kaspars; Manakova, Lena; Gražulis, Saulius; Matulis, Daumantas

Aryl-4,5-dihydro-1 H-pyrazole-1-carboxamide Derivatives Bearing a Sulfonamide Moiety Show Single-digit Nanomolar-to-Subnanomolar Inhibition Constants against the Tumor-associated Human Carbonic Anhydrases IX and XII

带有磺酰胺部分的芳基-4,5-二氢-1 H-吡唑-1-甲酰胺衍生物对肿瘤相关的人类碳酸酐酶 IX 和 XII 表现出个位数纳摩尔至亚纳摩尔抑制常数

Priya Hargunani, Nikhil Tadge, Mariangela Ceruso, Janis Leitans, Andris Kazaks, Kaspars Tars, Paola Gratteri, Claudiu T Supuran, Alessio Nocentini, Mrunmayee P Toraskar

Structures of plasmepsin II from Plasmodium falciparum in complex with two hydroxyethylamine-based inhibitors

恶性疟原虫疟原虫蛋白酶II与两种羟乙胺类抑制剂复合物的结构

Recacha, Rosario; Leitans, Janis; Akopjana, Inara; Aprupe, Lilija; Trapencieris, Peteris; Jaudzems, Kristaps; Jirgensons, Aigars; Tars, Kaspars