日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Di-meta-Substituted Fluorinated Benzenesulfonamides as Potent and Selective Anticancer Inhibitors of Carbonic Anhydrase IX and XII

二间位取代的氟化苯磺酰胺作为碳酸酐酶IX和XII的强效选择性抗癌抑制剂

Vaškevičius, Aivaras; Žvirblis, Mantas; Kurtenoka, Maija; Leitans, Janis; Manakova, Elena; Paketurytė-Latvė, Vaida; Kvietkauskaitė, Agnė; Kazaks, Andris; Eimonta, Vladislava; Čerepenkaitė, Kamilė; Kazokaitė-Adomaitienė, Justina; Mickevičiu̅tė, Aurelija; Juozapaitienė, Vaida; Tars, Kaspars; Gražulis, Saulius; Matulienė, Jurgita; Dudutienė, Virginija; Shubin, Kirill; Matulis, Daumantas; Zubrienė, Asta

Affinity and Selectivity of Protein-Ligand Recognition: A Minor Chemical Modification Changes Carbonic Anhydrase Binding Profile

蛋白质-配体识别的亲和力和选择性:微小的化学修饰改变碳酸酐酶的结合谱

Zakšauskas, Audrius; Paketurytė-Latvė, Vaida; Janku̅naitė, Alberta; Čapkauskaitė, Edita; Becart, Yann; Smirnov, Alexey; Pospíšilová, Klára; Leitans, Janis; Brynda, Jiří; Kazaks, Andris; Baranauskienė, Lina; Manakova, Elena; Gražulis, Saulius; Kairys, Visvaldas; Tars, Kaspars; Řezáčová, Pavlína; Matulis, Daumantas

Surface Functionalization of ITO for Dual-Mode Hypoxia-Associated Cancer Biomarker Detection.

用于双模式缺氧相关癌症生物标志物检测的ITO表面功能化

Zutis Edmunds, Paidere Gunita, Ruska Rihards, Freimanis Toms, Cipa Janis, Zalubovskis Raivis, Elksne Maira, Tars Kaspars, Kazaks Andris, Leitans Janis, Sarakovskis Anatolijs, Anspoks Andris

Targeted anticancer pre-vinylsulfone covalent inhibitors of carbonic anhydrase IX

靶向抗癌的碳酸酐酶IX前乙烯基砜共价抑制剂

Vaškevičius, Aivaras; Baronas, Denis; Leitans, Janis; Kvietkauskaitė, Agnė; Rukšėnaitė, Audronė; Manakova, Elena; Toleikis, Zigmantas; Kaupinis, Algirdas; Kazaks, Andris; Gedgaudas, Marius; Mickevičiūtė, Aurelija; Juozapaitienė, Vaida; Schiöth, Helgi B; Jaudzems, Kristaps; Valius, Mindaugas; Tars, Kaspars; Gražulis, Saulius; Meyer-Almes, Franz-Josef; Matulienė, Jurgita; Zubrienė, Asta; Dudutienė, Virginija; Matulis, Daumantas

From X-ray crystallographic structure to intrinsic thermodynamics of protein-ligand binding using carbonic anhydrase isozymes as a model system

以碳酸酐酶同工酶为模型体系,研究蛋白质-配体结合的X射线晶体结构及其内在热力学性质

Paketurytė-Latvė, Vaida; Smirnov, Alexey; Manakova, Elena; Baranauskiene, Lina; Petrauskas, Vytautas; Zubrienė, Asta; Matulienė, Jurgita; Dudutienė, Virginija; Čapkauskaitė, Edita; Zakšauskas, Audrius; Leitans, Janis; Gražulis, Saulius; Tars, Kaspars; Matulis, Daumantas

Isoform-Selective Enzyme Inhibitors by Exploring Pocket Size According to the Lock-and-Key Principle

基于锁钥原理,通过探索口袋大小来设计同工酶选择性酶抑制剂

Dudutienė, Virginija; Zubrienė, Asta; Kairys, Visvaldas; Smirnov, Alexey; Smirnovienė, Joana; Leitans, Janis; Kazaks, Andris; Tars, Kaspars; Manakova, Lena; Gražulis, Saulius; Matulis, Daumantas

Structures of plasmepsin II from Plasmodium falciparum in complex with two hydroxyethylamine-based inhibitors

恶性疟原虫疟原虫蛋白酶II与两种羟乙胺类抑制剂复合物的结构

Recacha, Rosario; Leitans, Janis; Akopjana, Inara; Aprupe, Lilija; Trapencieris, Peteris; Jaudzems, Kristaps; Jirgensons, Aigars; Tars, Kaspars