日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Advancing Structure Elucidation with a Flexible Multi-Spectral AI Model

利用灵活的多光谱人工智能模型推进结构解析

Priessner, Martin; Lewis, Richard J; Lemurell, Isak; Johansson, Magnus J; Goodman, JonathanM; Janet, Jon Paul; Tomberg, Anna

Conformational dynamics at the pre-miR-377 Dicer site governs selective small-molecule recognition

pre-miR-377 Dicer结合位点的构象动力学决定了其对小分子的选择性识别

Manigrasso, Jacopo; Mestdach, Emeline; Quaia, Riccardo; Dankova, Daniela; Bood, Mattias; Lemurell, Malin; Geschwindner, Stefan; Frolov, Andrey I; Disney, Matthew D; Hogner, Anders; Chi, Celestine N; Sala, Giuseppina La

Design of Bicyclic Peptide Tandems Mimicking the Homodimeric GDF15 Protein to Inhibit GDF15-GFRaL-RET Complex Cell Signaling

设计模拟同源二聚体GDF15蛋白的双环肽串联体以抑制GDF15-GFRaL-RET复合物细胞信号传导

Noisier, Anaïs F M; Sandmark, Jenny; Edfeldt, Fredrik; Backmark, Anna; Broddefalk, Johan; Wandzik, Joanna; Jurva, Ulrik; Ek, Margareta; Johansson, Carina A; Barlind, Louise; Gunnarsson, Jenny; Bigalke, Janna M; Xue, Yafeng; Frolov, Andrey I; Kankkonen, Cecilia; Roth, Robert G; Fritsch, Maria; Watcham, Sophie; van Rietschoten, Katerine; Mudd, Gemma E; Harrison, Helen; Chen, Liuhong; Skynner, Michael J; Craik, David J; Chankeshwara, Sunay V; Lemurell, Malin

Metabolic RNA labeling in non-engineered cells following spontaneous uptake of fluorescent nucleoside phosphate analogues

非工程细胞自发吸收荧光核苷磷酸类似物后进行代谢 RNA 标记

Pauline Pfeiffer, Jesper R Nilsson, Audrey Gallud, Tom Baladi, Hoang-Ngoan Le, Mattias Bood, Malin Lemurell, Anders Dahlén, Morten Grøtli, Elin K Esbjörner, L Marcus Wilhelmsson

A structure-specific small molecule inhibits a miRNA-200 family member precursor and reverses a type 2 diabetes phenotype

一种结构特异性小分子可抑制 miRNA-200 家族成员前体并逆转 2 型糖尿病表型

Hafeez S Haniff, Xiaohui Liu, Yuquan Tong, Samantha M Meyer, Laurent Knerr, Malin Lemurell, Daniel Abegg, Haruo Aikawa, Alexander Adibekian, Matthew D Disney

Fluorescent base analogues in gapmers enable stealth labeling of antisense oligonucleotide therapeutics

间隙体中的荧光碱基类似物可实现反义寡核苷酸疗法的隐形标记

Jesper R Nilsson, Tom Baladi, Audrey Gallud, Dženita Baždarević, Malin Lemurell, Elin K Esbjörner, L Marcus Wilhelmsson, Anders Dahlén

Design of a small molecule that stimulates vascular endothelial growth factor A enabled by screening RNA fold-small molecule interactions

通过筛选 RNA 折叠-小分子相互作用来设计刺激血管内皮生长因子 A 的小分子

Hafeez S Haniff, Laurent Knerr, Xiaohui Liu, Gogce Crynen, Jonas Boström, Daniel Abegg, Alexander Adibekian, Elizabeth Lekah, Kye Won Wang, Michael D Cameron, Ilyas Yildirim, Malin Lemurell, Matthew D Disney

A protein tertiary structure mimetic modulator of the Hippo signalling pathway

Hippo信号通路的一种蛋白质三级结构模拟调节剂

Hélène Adihou ,Ranganath Gopalakrishnan ,Tim Förster ,Stéphanie M Guéret ,Raphael Gasper ,Stefan Geschwindner ,Carmen Carrillo García ,Hacer Karatas ,Ajaybabu V Pobbati ,Mercedes Vazquez-Chantada ,Paul Davey ,Carola M Wassvik ,Jeremy Kah Sheng Pang ,Boon Seng Soh ,Wanjin Hong ,Elisabetta Chiarparin ,Dennis Schade ,Alleyn T Plowright ,Eric Valeur ,Malin Lemurell ,Tom N Grossmann ,Herbert Waldmann