日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Impact of SGLT2 Inhibitors on Preventing Heart Failure Hospitalizations in Colombian Patients With Uncontrolled Type 2 Diabetes Mellitus

SGLT2抑制剂对预防哥伦比亚未控制的2型糖尿病患者心力衰竭住院的影响

Vernaza Trujillo, David Alexander; Rojas Bautista, Lendy Yaneth; Ramirez Espinosa, Claudia Marcela; Sierra Castillo, Santiago; Corredor-Rengifo, David; Aristizabal Colorado, David; Abreu Lomba, Alin

Identification of PLCγ2 activators for the treatment of Alzheimer’s disease

鉴定用于治疗阿尔茨海默病的PLCγ2激活剂

Hawksley, J C; Clayton, Brent; Massey, Steven M; Chu, Shaoyou; Mason, Emily R; Bissel, Stephanie J; Bedford, Logan M; Rizzo, Stacey J Sukoff; Mesecar, Andrew D; Kaiser, Bridget L; Lendy, Emma K; Lamb, Bruce T; Palkowitz, Alan D; Richardson, Timothy I

Exploration of P1 and P4 modifications of nirmatrelvir: Design, synthesis, biological evaluation, and X-ray structural studies of SARS-CoV-2 Mpro inhibitors

探索尼尔马特雷韦的P1和P4修饰:SARS-CoV-2 Mpro抑制剂的设计、合成、生物学评价和X射线结构研究

Ghosh, Arun K; Yadav, Monika; Iddum, Satyanarayana; Ghazi, Somayeh; Lendy, Emma K; Jayashankar, Uttara; Beechboard, Sydney N; Takamatsu, Yuki; Hattori, Shin-Ichiro; Amano, Masayuki; Higashi-Kuwata, Nobuyo; Mitsuya, Hiroaki; Mesecar, Andrew D

Identification of PLCG2 activators for the treatment of Alzheimer’s disease

鉴定用于治疗阿尔茨海默病的PLCG2激活剂

Dang, Lei; Zhang, Chunbo; Su, Biru; Ning, Na; Huang, Qiuling; Zhou, Su; Wu, Meng; Ma, Wenqing; Wang, Man; Cui, Pengfei; Li, Yan; Wang, Shixuan; Clayton, Brent; Massey, Steven M; Beck, Daniel E; Putt, Karson S; Utsuki, Tada; Visvanathan, Ramya; Mesecar, Andrew D; Lendy, Emma K; Kaiser, Bridget L; Chu, Shaoyou; Mason, Emily R; Lamb, Bruce T; Palkowitz, Alan D; Richardson, Timothy I

A novel micellular fluorogenic substrate for quantitating the activity of 1-phosphatidylinositol 4,5-bisphosphate phosphodiesterase gamma (PLCγ) enzymes

一种用于定量测定 1-磷脂酰肌醇 4,5-二磷酸磷酸二酯酶 γ (PLCγ) 酶活性的新型细胞内荧光底物

Ramya Visvanathan ,Tadanobu Utsuki ,Daniel E Beck ,W Brent Clayton ,Emma Lendy ,Kuai-Lin Sun ,Yinghui Liu ,Kirk W Hering ,Andrew Mesecar ,Zhong-Yin Zhang ,Karson S Putt

Genetic variants of phospholipase C-γ2 alter the phenotype and function of microglia and confer differential risk for Alzheimer's disease

磷脂酶C-γ2的基因变异会改变小胶质细胞的表型和功能,并导致阿尔茨海默病风险的差异。

Andy P Tsai ,Chuanpeng Dong ,Peter Bor-Chian Lin ,Adrian L Oblak ,Gonzalo Viana Di Prisco ,Nian Wang ,Nicole Hajicek ,Adam J Carr ,Emma K Lendy ,Oliver Hahn ,Micaiah Atkins ,Aulden G Foltz ,Jheel Patel ,Guixiang Xu ,Miguel Moutinho ,John Sondek ,Qisheng Zhang ,Andrew D Mesecar ,Yunlong Liu ,Brady K Atwood ,Tony Wyss-Coray ,Kwangsik Nho ,Stephanie J Bissel ,Bruce T Lamb ,Gary E Landreth

Development of a sensitive microplate assay for characterizing RNA methyltransferase activity: Implications for epitranscriptomics and drug development.

开发一种灵敏的微孔板检测方法来表征 RNA 甲基转移酶活性:对表观转录组学和药物开发的影响

Mensah Isaiah K, Norvil Allison B, He Ming, Lendy Emma, Hjortland Nicole, Tan Hern, Pomerantz Richard T, Mesecar Andrew, Gowher Humaira

"There is a fear that you will be attacked just for the act of working in health": a survey of experiences of violence against healthcare in Colombia

“仅仅因为从事医疗工作,就担心会遭到攻击”:哥伦比亚医护人员遭受暴力侵害经历调查

Crawford, Katerina; Florez, Tatiana; Rodriguez, Mario; Cirado, Lendy; Read, Róisín; Haar, Rohini

A novel fluorogenic reporter substrate for 1-phosphatidylinositol 4,5-bisphosphate phosphodiesterase gamma-2 (PLCγ2): Application to high-throughput screening for activators to treat Alzheimer's disease

一种新型的1-磷脂酰肌醇4,5-二磷酸磷酸二酯酶γ-2 (PLCγ2)荧光报告底物:应用于阿尔茨海默病治疗激活剂的高通量筛选

Ramya Visvanathan ,Tadanobu Utsuki ,Daniel E Beck ,Emma Lendy ,Kuai-Lin Sun ,Yinghui Liu ,Kirk W Hering ,Andrew Mesecar ,Zhong-Yin Zhang ,Karson S Putt

A small molecule compound with an indole moiety inhibits the main protease of SARS-CoV-2 and blocks virus replication

含有吲哚部分的小分子化合物可抑制 SARS-CoV-2 的主要蛋白酶并阻止病毒复制

Shin-Ichiro Hattori, Nobuyo Higashi-Kuwata, Hironori Hayashi, Srinivasa Rao Allu, Jakka Raghavaiah, Haydar Bulut, Debananda Das, Brandon J Anson, Emma K Lendy, Yuki Takamatsu, Nobutoki Takamune, Naoki Kishimoto, Kazutaka Murayama, Kazuya Hasegawa, Mi Li, David A Davis, Eiichi N Kodama, Robert Yarcho