日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Targeting proteostasis in multiple myeloma through inhibition of LTK

通过抑制LTK靶向多发性骨髓瘤中的蛋白质稳态

Thea Kristin Våtsveen ,Mariaserena Giliberto ,Valgerdur Bjornsdottir ,Federica Centonze ,Andrej Besse ,Yannick Frey ,Sigrid S Skånland ,Anders Tveita ,Amin Alirezaylavasani ,John Franklin Imbery ,Kristine Misund ,Veronika Reiterer ,Muhammad Zahoor ,Christoph Driessen ,Lenka Besse ,Kjetil Tasken ,Fredrik H Schjesvold ,Hesso Farhan # ,Ludvig A Munthe #

Carfilzomib-specific proteasome β5/β2 inhibition drives cardiotoxicity via remodeling of protein homeostasis and the renin-angiotensin-system

卡非佐米特异性抑制蛋白酶体β5/β2通过重塑蛋白质稳态和肾素-血管紧张素系统而导致心脏毒性。

Max Mendez-Lopez ,Andrej Besse ,Christian Zuppinger ,Christian Perez-Shibayama ,Cristina Gil-Cruz ,Bogdan I Florea ,Angelina De Martin ,Mechthild Lütge ,Deborah Beckerova ,Simon Klimovic ,Xiang Zhou ,Leo Rasche ,Jan Pribyl ,Vladimir Rotrekl ,Burkhard Ludewig ,Herman S Overkleeft ,Lenka Besse ,Christoph Driessen

A replicating LCMV-based vaccine for the treatment of solid tumors

用于治疗实体肿瘤的复制型LCMV疫苗

Mette-Triin Purde, Jovana Cupovic, Yannick A Palmowski, Ahmad Makky, Sarah Schmidt, Alexander Rochwarger, Fabienne Hartmann, Felix Stemeseder, Alexander Lercher, Marie-Therese Abdou, David Bomze, Lenka Besse, Fiamma Berner, Thomas Tüting, Michael Hölzel, Andreas Bergthaler, Stefan Kochanek, Burkhard

HIV-protease inhibitors potentiate the activity of carfilzomib in triple-negative breast cancer

HIV 蛋白酶抑制剂增强卡非佐米在三阴性乳腺癌中的活性

Andrej Besse, Lenka Sedlarikova, Lorina Buechler, Marianne Kraus, Chieh-Hsiang Yang, Nicol Strakova, Karel Soucek, Jiri Navratil, Marek Svoboda, Alana L Welm, Markus Joerger, Christoph Driessen, Lenka Besse

Lysin (K)-specific demethylase 1 inhibition enhances proteasome inhibitor response and overcomes drug resistance in multiple myeloma

溶菌素 (K) 特异性去甲基化酶 1 抑制可增强蛋白酶体抑制剂反应并克服多发性骨髓瘤的耐药性

Cecilia Bandini, Elisabetta Mereu, Tina Paradzik, Maria Labrador, Monica Maccagno, Michela Cumerlato, Federico Oreglia, Lorenzo Prever, Veronica Manicardi, Elisa Taiana, Domenica Ronchetti, Mattia D'Agostino, Francesca Gay, Alessandra Larocca, Lenka Besse, Giorgio Roberto Merlo, Emilio Hirsch, Aless

The cytotoxic activity of carfilzomib together with nelfinavir is superior to the bortezomib/nelfinavir combination in non-small cell lung carcinoma

卡非佐米与奈非那韦联合治疗非小细胞肺癌的细胞毒活性优于硼替佐米/奈非那韦联合治疗

Lenka Besse, Marianne Kraus, Andrej Besse, Christoph Driessen, Ignazio Tarantino

The surfaceome of multiple myeloma cells suggests potential immunotherapeutic strategies and protein markers of drug resistance

多发性骨髓瘤细胞的表面组学研究提示了潜在的免疫治疗策略和耐药蛋白标志物。

Ian D Ferguson ,Bonell Patiño-Escobar ,Sami T Tuomivaara ,Yu-Hsiu T Lin ,Matthew A Nix ,Kevin K Leung ,Corynn Kasap ,Emilio Ramos ,Wilson Nieves Vasquez ,Alexis Talbot ,Martina Hale ,Akul Naik ,Audrey Kishishita ,Priya Choudhry ,Antonia Lopez-Girona ,Weili Miao ,Sandy W Wong ,Jeffrey L Wolf ,Thomas G Martin 3rd ,Nina Shah ,Scott Vandenberg ,Sonam Prakash ,Lenka Besse ,Christoph Driessen ,Avery D Posey Jr ,R Dyche Mullins ,Justin Eyquem ,James A Wells ,Arun P Wiita

Immunoproteasome Activity in Chronic Lymphocytic Leukemia as a Target of the Immunoproteasome-Selective Inhibitors

慢性淋巴细胞白血病中的免疫蛋白酶体活性作为免疫蛋白酶体选择性抑制剂的靶点

Andrej Besse, Marianne Kraus, Max Mendez-Lopez, Elmer Maurits, Herman S Overkleeft, Christoph Driessen, Lenka Besse

Treatment with HIV-Protease Inhibitor Nelfinavir Identifies Membrane Lipid Composition and Fluidity as a Therapeutic Target in Advanced Multiple Myeloma

使用 HIV 蛋白酶抑制剂奈非那韦治疗可确定膜脂质组成和流动性是晚期多发性骨髓瘤的治疗靶点

Lenka Besse #, Andrej Besse #, Sara C Stolze, Amin Sobh, Esther A Zaal, Alwin J van der Ham, Mario Ruiz, Santosh Phuyal, Lorina Büchler, Marc Sathianathan, Bogdan I Florea, Jan Borén, Marcus Ståhlman, Julia Huber, Arnold Bolomsky, Heinz Ludwig, J Thomas Hannich, Alex Loguinov, Bart Everts, Celia R B

Novel Peptide-drug Conjugate Melflufen Efficiently Eradicates Bortezomib-resistant Multiple Myeloma Cells Including Tumor-initiating Myeloma Progenitor Cells

新型肽类药物结合物美氟芬可有效消灭硼替佐米耐药多发性骨髓瘤细胞,包括肿瘤起始骨髓瘤祖细胞

Konstantin Byrgazov, Andrej Besse, Marianne Kraus, Ana Slipicevic, Fredrik Lehmann, Christoph Driessen, Lenka Besse