日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Overcoming Ligand Discovery Challenges: Developing Peptide-Based Tracers for SPSB2

克服配体发现挑战:开发用于 SPSB2 的基于肽的示踪剂

Lenz, Christopher; Elson, Lewis; Dopfer, Johannes; Farges, Frederic; Krämer, Andreas; Löhr, Frank; Müller, Susanne; Guéret, Stéphanie M; Waldmann, Herbert; Dötsch, Volker; Saxena, Krishna; Knapp, Stefan

Enantioselective protein affinity selection mass spectrometry (E-ASMS)

对映选择性蛋白质亲和力选择质谱法(E-ASMS)

Wang, Xiaoyun; Sun, Jianxian; Ahmad, Shabbir; Yang, Diwen; Li, Fengling; Chan, U Hang; Zeng, Hong; Simoben, Conrad V; Green, Stuart R; Silva, Madhushika; Houliston, Scott; Dong, Aiping; Bolotokova, Albina; Gibson, Elisa; Kutera, Maria; Ghiabi, Pegah; Kondratov, Ivan; Matviyuk, Tetiana; Chuprina, Alexander; Mavridi, Danai; Lenz, Christopher; Joerger, Andreas C; Brown, Benjamin D; Heath, Richard B; Yue, Wyatt W; Robbie, Lucy K; Beyett, Tyler S; Müller, Susanne; Knapp, Stefan; Owen, Dafydd R; Harding, Rachel; Schapira, Matthieu; Brown, Peter J; Santhakumar, Vijayaratnam; Ackloo, Suzanne; Arrowsmith, Cheryl H; Edwards, Aled M; Peng, Hui; Halabelian, Levon

Biochemical investigation of LC3/GABARAP-ligand interaction as an important quality measure for LC3/GABARAP-targeting small molecules: addendum to the guidelines (4th edition)

LC3/GABARAP-配体相互作用的生化研究作为LC3/GABARAP靶向小分子药物的重要质量指标:指南补充(第四版)

Schwalm, Martin P; Lenz, Christopher; Saxena, Krishna; Klionsky, Daniel J; Proschak, Ewgenij; Knapp, Stefan

Crystallographic fragment screening reveals ligand hotspots in TRIM21 PRY-SPRY domain.

晶体学片段筛选揭示了TRIM21 PRY-SPRY结构域中的配体热点

Kim Yeojin, Lučić Aleksandar, Lenz Christopher, Farges Frederic, Schwalm Martin P, Saxena Krishna, Hanke Thomas, Marples Peter G, Aschenbrenner Jasmin C, Fearon Daren, von Delft Frank, Krämer Andreas, Knapp Stefan

Un-LOK-ing a New Approach for Conformational Selective Targeting of STK10 (LOK)

针对 STK10 (LOK) 构象选择性靶向的新方法——解构 LOK

Dettenhöfer, Martina; Tandara, Laura Nadine; Amrhein, Jennifer Alisa; Kurz, Christian Georg; Schwalm, Martin Peter; Mensing, Theresa Elisabeth; Wahl, Laurenz Maximilian; Krämer, Andreas; Gerninghaus, Joshua; Lenz, Christopher; Elson, Lewis; Berger, Benedict-Tilman; Schröder, Martin; Saxena, Krishna; Müller, Susanne; Knapp, Stefan; Greco, Francesco Aleksy; Hanke, Thomas

Discovery of an exquisitely selective WDR5 chemical probe accelerated by a high-quality DEL-ML Hit

高质量的DEL-ML命中加速了极具选择性的WDR5化学探针的发现

Hoffmann, Lasse; Lenz, Christopher; Farges, Frederic; Kimani, Serah W; Dopfer, Johannes; Keller, Sabrina; Schwalm, Martin Peter; Holzmann, Hanna; Kraemer, Andreas; Dong, Aiping; Li, Fengling; Chau, Irene; Halabelian, Levon; Gstaiger, Matthias; Müller, Susanne; Knapp, Stefan; Němec, Václav

Enantioselective Protein Affinity Selection Mass Spectrometry (E-ASMS)

对映选择性蛋白质亲和力选择质谱法 (E-ASMS)

Wang, Xiaoyun; Sun, Jianxian; Ahmad, Shabbir; Yang, Diwen; Li, Fengling; Chan, U Hang; Zeng, Hong; Simoben, Conrad V; Green, Stuart R; Silva, Madhushika; Houliston, Scott; Dong, Aiping; Bolotokova, Albina; Gibson, Elisa; Kutera, Maria; Ghiabi, Pegah; Kondratov, Ivan; Matviyuk, Tetiana; Chuprina, Alexander; Mavridi, Danai; Lenz, Christopher; Joerger, Andreas C; Brown, Benjamin D; Heath, Richard B; Yue, Wyatt W; Robbie, Lucy K; Beyett, Tyler S; Müller, Susanne; Knapp, Stefan; Harding, Rachel; Schapira, Matthieu; Brown, Peter J; Santhakumar, Vijayaratnam; Ackloo, Suzanne; Arrowsmith, Cheryl H; Edwards, Aled M; Peng, Hui; Halabelian, Levon

Back-Pocket Optimization of 2-Aminopyrimidine-Based Macrocycles Leads to Potent EPHA2/GAK Kinase Inhibitors.

2-氨基嘧啶基大环化合物的后口袋优化可得到强效的EPHA2/GAK激酶抑制剂

Gerninghaus Joshua, Zhubi Rezart, Krämer Andreas, Karim Marwah, Tran Do Hoang Nhu, Joerger Andreas C, Schreiber Christian, Berger Lena M, Berger Benedict-Tilman, Ehret Theresa A L, Elson Lewis, Lenz Christopher, Saxena Krishna, Müller Susanne, Einav Shirit, Knapp Stefan, Hanke Thomas

Non-Adherence to Pain Medication Increases Risk of Postoperative Frozen Shoulder

不遵医嘱服用止痛药会增加术后肩周炎的风险

Niehaus, Richard; Urbanschitz, Lukas; Schumann, Jakob; Lenz, Christopher G; Frank, Florian A; Ehrendorfer, Stefan; Eid, Karim

A114 SYSTEMATIC REVIEW AND META-ANALYSIS: ENDOSCOPIC AND HISTOLOGIC PLACEBO RATES IN INDUCTION AND MAINTENANCE TRIALS OF ULCERATIVE COLITIS

A114 系统评价和荟萃分析:溃疡性结肠炎诱导和维持治疗试验中的内镜和组织学安慰剂率

Rashed, Reem; Valcheva, Rosica; Dieleman, Levinus A; Pattisapu, Naveen; Huang, Dave; Porter, Giselle M; Owhonda, Rebisi; Charlton, Timothy; Gross, Christopher E; Thordarson, David; Metzger, Melodie; Yammine, Kaissar; Sayegh, George E; ElAlam, Anthony; Jamaleddine, Youssef; Mouawad, Joseph; Assi, Chahine; Lui, Chun Wai; Loureiro, Rui CV; Malhotra, Karan; Allen, Nicholas; Aitchison, Alexandra Hunter; Bagheri, Kian; Guardino, Nicholas; Abar, Bijan; Anastasio, Albert T; Adams, Samuel; Meldau, Jason; LeDuc, Ryan; Havey, Robert; Muriuki, Muturi; Kaczmarz, Nadia; Schiff, Adam; Ravn-Boess, Niklas; Bhowmick, Nainita; Hattori, Takamitsu; Prakash, Varsha; Stephan, Gabriele; Frenster, Joshua; Bready, Devin; Lawson, Christopher; Wilcox, Jordan; Placantonakis, Dimitris; Trudil, D; Loomis, L; MacAry, P; Almond, G; Smallfield, Jessica; Dahmer, Payton L; Harrison, Olivia; Jones, Cassandra K; Ravn-Boess, Niklas; Bhowmick, Nainita; Hattori, Takamitsu; Corrado, Alexis; Koide, Akiko; Karimkhan, Afreen; Koide, Shohei; Park, Christopher; Placantonakis, Dimitris; Cornelius, Canon C; Daniels, Joseph; Garcia, Hugo C; Warner, Stephen J; Lenz, Christopher G; Raith, Constance; Urbanschitz, Lukas; Tondelli, Timo O; Eid, Karim; Niehaus, Richard; Hodel, Sandro; Teramoto, Atsushi; Murahashi, Yasutaka; Shoji, Hiroaki; Kamiya, Tomoaki; Watanabe, Kota; Yamashita, Toshihiko; Kukowski, Nathan; Wilson, Jacob M; Bariteau, Jason T; Staley, Christopher A; Ashkani-Esfahani, Soheil; Lubberts, Bart; Bhimani, Rohan; DiGiovanni, Christopher W; Ma, C; Guizzetti, L; Panaccione, R; Fedorak, R; Parker, C E; Nguyen, T; Khanna, R; Feagan, B G; Jairath, V