日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of small molecule modulators of the thin filament that alter the contractile profile in a hypertrophic cardiomyopathy engineered tissue model

在肥厚型心肌病工程组织模型中,发现了能够改变细丝收缩特性的小分子调节剂

Sommese, Ruth F; Levi, Samuel M; Brown, Janice; Polivkova, Jana; Byrnes, Laura J; Kue, Richard; Damilano, Federico; Hua, Wenyi; Boehm, Markus; Dushin, Elizabeth; Filipski, Kevin J; Kormos, Bethany L; Li, Qifang; Miller, Russell; Ogilvie, Kevin; Ridgway, Noelle; Smith, Aaron C; Stansfield, John C; Wang, Yang; Withka, Jane; Zhang, Hui; Griffith, David A; Ward, Jessica

Unifying Catalysis Framework to Dissect Proteasomal Degradation Paradigms

统一催化框架以剖析蛋白酶体降解范式

Rodriguez-Rivera, Frances P; Levi, Samuel M

Discovery of Diaminopyrimidine Carboxamide HPK1 Inhibitors as Preclinical Immunotherapy Tool Compounds

二氨基嘧啶羧酰胺类HPK1抑制剂作为临床前免疫治疗工具化合物的发现

Vara, Brandon A; Levi, Samuel M; Achab, Abdelghani; Candito, David A; Fradera, Xavier; Lesburg, Charles A; Kawamura, Shuhei; Lacey, Brian M; Lim, Jongwon; Methot, Joey L; Xu, Zangwei; Xu, Haiyan; Smith, Dustin M; Piesvaux, Jennifer A; Miller, J Richard; Bittinger, Mark; Ranganath, Sheila H; Bennett, David J; DiMauro, Erin F; Pasternak, Alexander

Highly Selective β-Mannosylations and β-Rhamnosylations Catalyzed by Bis-thiourea

双硫脲催化的高选择性β-甘露糖基化和β-鼠李糖基化

Li, Qiuhan; Levi, Samuel M; Jacobsen, Eric N

Catalytic activation of glycosyl phosphates for stereoselective coupling reactions

糖基磷酸酯的催化活化用于立体选择性偶联反应

Levi, Samuel M; Li, Qiuhan; Rötheli, Andreas R; Jacobsen, Eric N

Autophagy Inhibition Enhances Sunitinib Efficacy in Clear Cell Ovarian Carcinoma

自噬抑制增强舒尼替尼在透明细胞卵巢癌中的疗效

DeVorkin, Lindsay; Hattersley, Matthew; Kim, Paul; Ries, Jenna; Spowart, Jaeline; Anglesio, Michael S; Levi, Samuel M; Huntsman, David G; Amaravadi, Ravi K; Winkler, Jeffrey D; Tinker, Anna V; Lum, Julian J

Autophagy gene Atg16L1 prevents lethal T cell alloreactivity mediated by dendritic cells.

自噬基因Atg16L1可阻止树突状细胞介导的致命性T细胞同种异体反应

Hubbard-Lucey Vanessa M, Shono Yusuke, Maurer Katie, West Mallory L, Singer Natalie V, Ziegler Carly G K, Lezcano Cecilia, Motta Ana Carolina Fragoso, Schmid Karin, Levi Samuel M, Murphy George F, Liu Chen, Winkler Jeffrey D, Amaravadi Ravi K, Rogler Gerhard, Dickinson Anne M, Holler Ernst, van den Brink Marcel R M, Cadwell Ken

Autophagy inhibitor Lys05 has single-agent antitumor activity and reproduces the phenotype of a genetic autophagy deficiency

自噬抑制剂Lys05具有单药抗肿瘤活性,并能重现遗传性自噬缺陷的表型。

McAfee, Quentin; Zhang, Zhihui; Samanta, Arabinda; Levi, Samuel M; Ma, Xiao-Hong; Piao, Shengfu; Lynch, John P; Uehara, Takeshi; Sepulveda, Antonia R; Davis, Lisa E; Winkler, Jeffrey D; Amaravadi, Ravi K