日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structures of partially occupied hetero-tetramers provide insight into kainate receptor activation and desensitization

部分占据的异源四聚体的结构为红藻氨酸受体的激活和脱敏提供了见解

Khanra, Nandish K; Strauss, Alexa; Moreno Wasielewski, Laura; Lenze, Sophie; Meyerson, Joel; Reiner, Andreas; Levitz, Joshua

TrkB/mGluR5 cross-talk underlies a synaptic metaplasticity mechanism of ketamine

TrkB/mGluR5 相互作用是氯胺酮突触元可塑性机制的基础。

Arefin, Anisul; Kim, Jihye; Chakraborty, Manas Pratim; Martinelli, Silvia; Bai, Betty; Lee, Francis S; Levitz, Joshua

Developing HaloTag and SNAP-Tag Chemical Inducers of Dimerization to Probe Receptor Oligomerization and Downstream Signaling

开发 HaloTag 和 SNAP-Tag 二聚化化学诱导剂以探测受体寡聚化和下游信号传导

Trumpp, Michael; Gatin-Fraudet, Blaise; Bruckmann, Kjell; Burdzinski, Wiktor; Roßmann, Kilian; Levitz, Joshua; Knaus, Petra; Jatzlau, Jerome; Broichhagen, Johannes

Projection-targeted photopharmacology reveals distinct anxiolytic roles for presynaptic mGluR2 in prefrontal- and insula-amygdala synapses.

投射靶向光药理学揭示了前额叶和岛叶杏仁核突触中突触前 mGluR2 的独特抗焦虑作用

Munguba Hermany, Srivastava Ipsit, Gutzeit Vanessa A, Singh Ashna, Vijay Akshara, Kristt Melanie, Arefin Anisul, Thukral Sonal, Broichhagen Johannes, Stujenske Joseph M, Liston Conor, Levitz Joshua

The accessory protein MRAP2 directly interacts with melanocortin-3 receptor to enhance signaling.

辅助蛋白 MRAP2 直接与黑皮质素-3 受体相互作用,增强信号传导。

Jamaluddin Aqfan, Wyatt Rachael A, Lee Joon, Dowsett Georgina K C, Tadross John A, Broichhagen Johannes, Yeo Giles S H, Levitz Joshua, Gorvin Caroline M

Red and far-red cleavable fluorescent dyes for self-labelling enzyme protein tagging and interrogation of GPCR co-internalization

用于酶蛋白自标记和GPCR共内化检测的红色和远红外可裂解荧光染料

Roßmann, Kilian; Birke, Ramona; Levitz, Joshua; Jones, Ben; Broichhagen, Johannes

An opioid efficacy switch for reversible optical control of peripheral analgesia

用于可逆性光学控制外周镇痛的阿片类药物疗效开关

Posa, Luca; Romano, Giovanna; Ji, Xiang; Khan, Saif; Paz, Bruno Matos; Han, Gye Won; Nazarova, Antonina L; Zaidi, Saheem A; Ranjbar, Mohsen; Pleil, Kristen; Katritch, Vsevolod; Gati, Cornelius; Trauner, Dirk; Levitz, Joshua

Structural Diversity and Dynamics of Metabotropic Glutamate Receptor/Beta-Arrestin Coupling

代谢型谷氨酸受体/β-arrestin偶联的结构多样性和动力学

Marx, Dagan C; Huynh, Kevin; Gonzalez-Hernandez, Alberto J; Strauss, Alexa; Rico, Carlos; Siepe, Dirk; Gallo, Pamela N; Lee, Joon; Moshtaghin, Sheida Sharghi; Arefin, Anisul; Weber, Willem F; Broichhagen, Johannes; Eliezer, David; Kalocsay, Marian; Khelashvili, George; Levitz, Joshua

MRAP2 potentiates GPCR signaling by conserved mechanisms that are disrupted by obesity-associated genetic variants.

MRAP2 通过保守机制增强 GPCR 信号传导,而肥胖相关的基因变异会破坏这些机制。

Jamaluddin Aqfan, Wyatt Rachael A, Broichhagen Johannes, Levitz Joshua, Gorvin Caroline M

Author Correction: Combined small-molecule treatment accelerates maturation of human pluripotent stem cell-derived neurons

作者更正:联合小分子治疗加速人类多能干细胞衍生神经元的成熟

Hergenreder, Emiliano; Minotti, Andrew P; Zorina, Yana; Oberst, Polina; Zhao, Zeping; Munguba, Hermany; Calder, Elizabeth L; Baggiolini, Arianna; Walsh, Ryan M; Liston, Conor; Levitz, Joshua; Garippa, Ralph; Chen, Shuibing; Ciceri, Gabriele; Studer, Lorenz