日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structural optimization of drug molecules with incrementally trained language models

利用增量训练的语言模型进行药物分子结构优化

Hörmann, Tim; Mayer, Domenic; Lewandowski, Max; Hunklinger, Andrea; Wein, Thomas; Merk, Daniel

Click. Screen. Degrade. A Miniaturized D2B Workflow for Rapid PROTAC Discovery

点击。屏幕。降级。用于快速 PROTAC 发现的微型化 D2B 工作流程

Mitrović, Marko; Greco, Francesco Aleksy; García, Yiliam Cruz; Lučić, Aleksandar; Hoffmann, Lasse; Chander, Rohit; Schönfeld, Julia; Liebisch, Nick; Sivashanmugam, Saran Aswathaman; Schwalm, Martin Peter; Egner, Markus; Lewandowski, Max; Merk, Daniel; Morasch, Viktoria; Wolf, Elmar; Müller, Susanne; Hanke, Thomas; Proschak, Ewgenij; Hiesinger, Kerstin; Knapp, Stefan

A Nurr1 Agonist Derived from the Natural Ligand DHI Induces Neuroprotective Gene Expression.

源自天然配体DHI的Nurr1激动剂可诱导神经保护基因表达

Egner Markus, Busch Romy, López-García Úrsula, Lewandowski Max, Höfner Georg, Wein Thomas, Marschner Julian A, Merk Daniel

Comparative Evaluation and Profiling of Chemical Tools for the Nuclear Hormone Receptor Family 2.

核激素受体家族 2 化学工具的比较评价和分析

Lewandowski Max, Busch Romy, Marschner Julian A, Merk Daniel