日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Sevabertinib, a Reversible HER2 Inhibitor with Activity in Lung Cancer

塞伐替尼,一种对肺癌有效的可逆性HER2抑制剂

Siegel, Franziska; Siegel, Stephan; Kotýnková, Kristýna; Karsli Uzunbas, Gizem; Korr, Daniel; Tomono, Haruna; Andersen, Sawyer; Denney, Daniel; Berger, Markus; Schulze, Volker K; Lewis, Timothy A; Kaplan, Bethany; Golfier, Sven; Mortier, Jérémie; Hillig, Roman C; Boemer, Ulf; Petersen, Kirstin; Eis, Knut; Williams, Sybil; Rüttinger, Dominik; Cherniack, Andrew D; Loong, Herbert H; Goto, Koichi; Grassi, Paolo; Meyerson, Matthew; Greulich, Heidi

Discovery of BAY 2666605, a Molecular Glue for PDE3A and SLFN12

BAY 2666605 的发现,一种 PDE3A 和 SLFN12 的分子胶

Lewis, Timothy A; Ellermann, Manuel; Kopitz, Charlotte; Lange, Martin; de Waal, Luc; Wu, Xiaoyun; Tersteegen, Adrian; Denner, Karsten; Lienau, Philip; Kaulfuss, Stefan; Goldoni, Silvia; Meyerson, Matthew; Greulich, Heidi; Gradl, Stefan N

NIAID workshop on T cell technologies

美国国家过敏症和传染病研究所 (NIAID) T 细胞技术研讨会

Gondré-Lewis, Timothy A; Jiang, Chao; Ford, Mandy L; Koelle, David M; Sette, Alessandro; Shalek, Alex K; Thomas, Paul G

The Opioid Epidemic: a Crisis Disproportionately Impacting Black Americans and Urban Communities

阿片类药物危机:对非裔美国人和城市社区的影响尤为严重

Gondré-Lewis, Marjorie C; Abijo, Tomilowo; Gondré-Lewis, Timothy A

Correction: Mechanistic insights into cancer cell killing through interaction of phosphodiesterase 3A and schlafen family member 12

更正:磷酸二酯酶 3A 与 Schlafen 家族成员 12 相互作用导致癌细胞死亡的机制研究

Wu, Xiaoyun; Schnitzler, Gavin R; Gao, Galen F; Diamond, Brett; Baker, Andrew R; Kaplan, Bethany; Williamson, Kaylyn; Westlake, Lindsay; Lorrey, Selena; Lewis, Timothy A; Garvie, Colin W; Lange, Martin; Hayat, Sikander; Seidel, Henrik; Doench, John; Cherniack, Andrew D; Kopitz, Charlotte; Meyerson, Matthew; Greulich, Heidi

Diversity-oriented synthesis yields novel multistage antimalarial inhibitors.

多样性导向合成产生新型多阶段抗疟疾抑制剂

Kato Nobutaka, Comer Eamon, Sakata-Kato Tomoyo, Sharma Arvind, Sharma Manmohan, Maetani Micah, Bastien Jessica, Brancucci Nicolas M, Bittker Joshua A, Corey Victoria, Clarke David, Derbyshire Emily R, Dornan Gillian L, Duffy Sandra, Eckley Sean, Itoe Maurice A, Koolen Karin M J, Lewis Timothy A, Lui Ping S, Lukens Amanda K, Lund Emily, March Sandra, Meibalan Elamaran, Meier Bennett C, McPhail Jacob A, Mitasev Branko, Moss Eli L, Sayes Morgane, Van Gessel Yvonne, Wawer Mathias J, Yoshinaga Takashi, Zeeman Anne-Marie, Avery Vicky M, Bhatia Sangeeta N, Burke John E, Catteruccia Flaminia, Clardy Jon C, Clemons Paul A, Dechering Koen J, Duvall Jeremy R, Foley Michael A, Gusovsky Fabian, Kocken Clemens H M, Marti Matthias, Morningstar Marshall L, Munoz Benito, Neafsey Daniel E, Sharma Amit, Winzeler Elizabeth A, Wirth Dyann F, Scherer Christina A, Schreiber Stuart L

Dilazep analogues for the study of equilibrative nucleoside transporters 1 and 2 (ENT1 and ENT2)

用于研究平衡型核苷转运体 1 和 2 (ENT1 和 ENT2) 的地拉泽普类似物

Playa, Hilaire; Lewis, Timothy A; Ting, Amal; Suh, Byung-Chul; Muñoz, Benito; Matuza, Robert; Passer, Brent J; Schreiber, Stuart L; Buolamwini, John K

Identification of regulators of polyploidization presents therapeutic targets for treatment of AMKL

鉴定多倍体化调控因子可为治疗急性髓系白血病(AMKL)提供治疗靶点。

Wen, Qiang; Goldenson, Benjamin; Silver, Serena J; Schenone, Monica; Dancik, Vlado; Huang, Zan; Wang, Ling-Zhi; Lewis, Timothy A; An, W Frank; Li, Xiaoyu; Bray, Mark-Anthony; Thiollier, Clarisse; Diebold, Lauren; Gilles, Laure; Vokes, Martha S; Moore, Christopher B; Bliss-Moreau, Meghan; Verplank, Lynn; Tolliday, Nicola J; Mishra, Rama; Vemula, Sasidhar; Shi, Jianjian; Wei, Lei; Kapur, Reuben; Lopez, Cécile K; Gerby, Bastien; Ballerini, Paola; Pflumio, Francoise; Gilliland, D Gary; Goldberg, Liat; Birger, Yehudit; Izraeli, Shai; Gamis, Alan S; Smith, Franklin O; Woods, William G; Taub, Jeffrey; Scherer, Christina A; Bradner, James E; Goh, Boon-Cher; Mercher, Thomas; Carpenter, Anne E; Gould, Robert J; Clemons, Paul A; Carr, Steven A; Root, David E; Schreiber, Stuart L; Stern, Andrew M; Crispino, John D

Inhibition of histone deacetylase 3 protects beta cells from cytokine-induced apoptosis

抑制组蛋白去乙酰化酶3可保护β细胞免受细胞因子诱导的细胞凋亡

Chou, Danny Hung-Chieh; Holson, Edward B; Wagner, Florence F; Tang, Alicia J; Maglathlin, Rebecca L; Lewis, Timothy A; Schreiber, Stuart L; Wagner, Bridget K

Rho kinase regulates the survival and transformation of cells bearing oncogenic forms of KIT, FLT3, and BCR-ABL

Rho激酶调控携带致癌型KIT、FLT3和BCR-ABL的细胞的存活和转化。

Mali, Raghuveer Singh; Ramdas, Baskar; Ma, Peilin; Shi, Jianjian; Munugalavadla, Veerendra; Sims, Emily; Wei, Lei; Vemula, Sasidhar; Nabinger, Sarah C; Goodwin, Charles B; Chan, Rebecca J; Traina, Fabiola; Visconte, Valeria; Tiu, Ramon V; Lewis, Timothy A; Stern, Andrew M; Wen, Qiang; Crispino, John D; Boswell, H Scott; Kapur, Reuben