日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Type II kinase inhibitors that target Parkinson's disease-associated LRRK2

靶向帕金森病相关LRRK2的II型激酶抑制剂

Nicolai D Raig ,Katherine J Surridge ,Marta Sanz-Murillo ,Verena Dederer ,Andreas Krämer ,Martin P Schwalm ,Nicholas M Lattal ,Lewis Elson ,Deep Chatterjee ,Sebastian Mathea ,Thomas Hanke ,Andres E Leschziner ,Samara L Reck-Peterson ,Stefan Knapp

Covalent Targeting Leads to the Development of a LIMK1 Isoform-Selective Inhibitor

共价靶向导致LIMK1亚型选择性抑制剂的开发

Sebastian Mandel ,Thomas Hanke ,Niall Prendiville ,María Baena-Nuevo ,Lena Marie Berger ,Frederic Farges ,Martin Peter Schwalm ,Benedict-Tilman Berger ,Andreas Kraemer ,Lewis Elson ,Hayuningbudi Saraswati ,Kamal R Abdul Azeez ,Verena Dederer ,Sebastian Mathea ,Ana Corrionero ,Patricia Alfonso ,Sabrina Keller ,Matthias Gstaiger ,Daniela S Krause ,Susanne Müller ,Sandra Röhm ,Stefan Knapp

Chemogenomics for steroid hormone receptors (NR3)

类固醇激素受体(NR3)化学基因组学

Espen Schallmayer, Laura Isigkeit, Lewis Elson, Susanne Müller, Stefan Knapp, Julian A Marschner, Daniel Merk

Type-II kinase inhibitors that target Parkinson's Disease-associated LRRK2

针对帕金森病相关 LRRK2 的 II 型激酶抑制剂

Nicolai D Raig, Katherine J Surridge, Marta Sanz-Murillo, Verena Dederer, Andreas Krämer, Martin P Schwalm, Lewis Elson, Deep Chatterjee, Sebastian Mathea, Thomas Hanke, Andres E Leschziner, Samara L Reck-Peterson, Stefan Knapp

Chemogenomics for NR1 nuclear hormone receptors

NR1 核激素受体化学基因组学

Laura Isigkeit #, Espen Schallmayer #, Romy Busch, Lorene Brunello, Amelie Menge, Lewis Elson, Susanne Müller, Stefan Knapp, Alexandra Stolz, Julian A Marschner, Daniel Merk

Back-pocket optimization of 2-aminopyrimidine-based macrocycles leads to potent dual EPHA2/GAK kinase inhibitors with antiviral activity

对 2-氨基嘧啶大环化合物进行后袋优化,可得到具有抗病毒活性的强效双重 EPHA2/GAK 激酶抑制剂

Joshua Gerninghaus, Rezart Zhubi, Andreas Krämer, Marwah Karim, Do Hoang Nhu Tran, Andreas C Joerger, Christian Schreiber, Lena M Berger, Benedict-Tilman Berger, Theresa A L Ehret, Lewis Elson, Christopher Lenz, Krishna Saxena, Susanne Müller, Shirit Einav, Stefan Knapp, Thomas Hanke

Discovery of 3-Amino-1 H-pyrazole-Based Kinase Inhibitors to Illuminate the Understudied PCTAIRE Family

发现基于 3-氨基-1 H-吡唑的激酶抑制剂,为尚未深入研究的 PCTAIRE 家族提供启示

Jennifer Alisa Amrhein, Lena Marie Berger, Amelie Tjaden, Andreas Krämer, Lewis Elson, Tuomas Tolvanen, Daniel Martinez-Molina, Astrid Kaiser, Manfred Schubert-Zsilavecz, Susanne Müller, Stefan Knapp, Thomas Hanke