日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

OICR-41103 as a chemical probe for the DCAF1 WD40 domain.

OICR-41103 作为 DCAF1 WD40 结构域的化学探针

Kimani Serah W, Noureldin Mahmoud, Wilson Brian, Hoffer Laurent, Green Stuart R, Szewczyk Magdalena M, González-Álvarez Héctor, Mohammed Mohammed, Chan Manuel, Krausser Chiara, Li Alice Shi Ming, Hajian Taraneh, Tucker Sarah, Joshi Dhananjay, Saraon Punit, Thériault Brigitte, Kim Ji Sup, Santhakumar Vijayaratnam, Loppnau Peter, Li Yanjun, Seitova Almagul, Dong Aiping, Kiyota Taira, Hammann Tobias, Gehrtz Paul, Patel Bhashant, Rathod Vaibhavi, Vala Anand, Rout Bhimsen, Jagodra Paras, Brown Peter J, Aman Ahmed, Ramnauth Jailall, Poda Gennady, Uehling David, Arrowsmith Cheryl H, Barsyte-Lovejoy Dalia, Marcellus Richard, Ackloo Suzanne, Mamai Ahmed, Al-Awar Rima, Halabelian Levon

Rational Design of Highly Potent SARS-CoV-2 nsp14 Methyltransferase Inhibitors

高效SARS-CoV-2 nsp14甲基转移酶抑制剂的合理设计

Štefek, Milan; Chalupská, Dominika; Chalupský, Karel; Zgarbová, Michala; Dvořáková, Alexandra; Krafčíková, Petra; Li, Alice Shi Ming; Šála, Michal; Dejmek, Milan; Otava, Tomáš; Chaloupecká, Ema; Kozák, Jaroslav; Kozic, Ján; Vedadi, Masoud; Weber, Jan; Mertlíková-Kaiserová, Helena; Nencka, Radim

Discovery of a Druggable, Cryptic Pocket in SARS-CoV-2 nsp16 Using Allosteric Inhibitors

利用变构抑制剂发现SARS-CoV-2 nsp16中一个可成药的隐蔽口袋

Inniss, Nicole L; Kozic, Ján; Li, Fengling; Rosas-Lemus, Monica; Minasov, George; Rybáček, Jiří; Zhu, Yingjie; Pohl, Radek; Shuvalova, Ludmilla; Rulíšek, Lubomír; Brunzelle, Joseph S; Bednárová, Lucie; Štefek, Milan; Kormaník, Ján Michael; Andris, Erik; Šebestík, Jaroslav; Li, Alice Shi Ming; Brown, Peter J; Schmitz, Uli; Saikatendu, Kumar; Chang, Edcon; Nencka, Radim; Vedadi, Masoud; Satchell, Karla J F

Design and synthesis of naturally-inspired SARS-CoV-2 inhibitors

天然SARS-CoV-2抑制剂的设计与合成

Hassan, Haitham; Chiavaralli, Jeanne; Hassan, Afnan; Bedda, Loay; Krischuns, Tim; Chen, Kuang-Yu; Li, Alice Shi Ming; Delpal, Adrien; Decroly, Etienne; Vedadi, Masoud; Naffakh, Nadia; Agou, Fabrice; Mallart, Sergio; Arafa, Reem K; Arimondo, Paola B