日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of clofibric acid as a SYVN1 ligand for PROTAC development

氯贝酸作为SYVN1配体在PROTAC开发中的鉴定

Warren, Julia; Munakala, Anandarao; Zientek, Keith D; Kim, Kilsun; Wilmarth, Phil A; Reddy, Ashok P; Li, Bingbing X; Xiao, Xiangshu

Discovery of peptidomimetic inhibitors of CREB/CBP by targeting hydrophobic grooves on the surface of the CBP KIX domain

通过靶向CBP KIX结构域表面的疏水沟槽,发现CREB/CBP的肽模拟抑制剂。

Huang, Bo; Gregory-Lott, Emily; Li, Bingbing X; Tran, Timothy H; Li, Sihao; Xue, Menglin; Wang, Shaohui; Asokan, Anabanadam; Shen, Ning; Sun, Xingming; Cao, Chuanhai; Xiao, Xiangshu; Daughdrill, Gary; Cai, Jianfeng

Recognition of the CREB-Binding Protein/Mixed Lineage Leukemia Interface by Sulfonyl-γ-AApeptides: Beyond Mimicry of Mixed Lineage Leukemia

磺酰-γ-AA肽对CREB结合蛋白/混合谱系白血病界面的识别:超越混合谱系白血病的模拟

Huang, Bo; Wang, Minghui; Gregory-Lott, Emily; Li, Bingbing X; Win, Yu Yu; Shen, Ning; Chen, Jianyu; Li, Sihao; Cao, Chuanhai; Xiao, Xiangshu; Daughdrill, Gary W; Cai, Jianfeng

Establishing preclinical models for clear cell sarcoma of soft tissue

建立软组织透明细胞肉瘤的临床前模型

Li, Bingbing X; Piesner, Jake

Design, synthesis and evaluation of clickable photoaffinity probes for nuclear lamins

核纤层蛋白可点击光亲和探针的设计、合成和评价

Warren, Julia; Wang, Jian; Li, Bingbing X; Xiao, Xiangshu

Dual Labeling of Newly Synthesized Proteins and Existing Proteins Using (CG)-SLENP.

利用 (CG)-SLENP 对新合成蛋白质和现有蛋白质进行双重标记

Li Bingbing X, Xiao Xiangshu

(CG)-SLENP: A Chemical Genetics Strategy To Selectively Label Existing Proteins and Newly Synthesized Proteins.

(CG)-SLENP:一种选择性标记现有蛋白质和新合成蛋白质的化学遗传学策略

Wang Jian, Chao Bo, Piesner Jake, Kelly Felice, Petrie Stefanie Kaech, Xiao Xiangshu, Li Bingbing X

Mechanistic insights into the activation of ester prodrugs of 666-15

对 666-15 酯类前药活化的机制研究

Xie, Fuchun; Martín-Acosta, Pedro; Li, Bingbing X; Xiao, Xiangshu

A suite of bioassays to evaluate CREB inhibitors

一套用于评估 CREB 抑制剂的生物测定方法

Li, Bingbing X; Xiao, Xiangshu

Identification of lamins as the molecular targets of LBL1 using a clickable photoaffinity probe.

利用可点击光亲和探针鉴定层粘蛋白为 LBL1 的分子靶标

Xiao Xiangshu, Li Bingbing X