日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Exploring the target scope of KEAP1 E3 ligase-based PROTACs

探索基于 KEAP1 E3 连接酶的 PROTAC 的靶标范围

Guangyan Du, Jie Jiang, Nathaniel J Henning, Nozhat Safaee, Eriko Koide, Radosław P Nowak, Katherine A Donovan, Hojong Yoon, Inchul You, Hong Yue, Nicholas A Eleuteri, Zhixiang He, Zhengnian Li, Hubert T Huang, Jianwei Che, Behnam Nabet, Tinghu Zhang, Eric S Fischer, Nathanael S Gray

Potency- and Selectivity-Enhancing Mutations of Conotoxins for Nicotinic Acetylcholine Receptors Can Be Predicted Using Accurate Free-Energy Calculations

利用精确的自由能计算可以预测芋螺毒素对尼古丁乙酰胆碱受体的效力和选择性增强突变

Katz, Dana; DiMattia, Michael A; Sindhikara, Dan; Li, Hubert; Abraham, Nikita; Leffler, Abba E

EPHA2 mutations with oncogenic characteristics in squamous cell lung cancer and malignant pleural mesothelioma

EPHA2 突变在鳞状细胞肺癌和恶性胸膜间皮瘤中具有致癌特征

Tan, Yi-Hung Carol; Srivastava, Saumya; Won, Brian M; Kanteti, Rajani; Arif, Qudsia; Husain, Aliya N; Li, Hubert; Vigneswaran, Wickii T; Pang, Ka-Ming; Kulkarni, Prakash; Sattler, Martin; Vaidehi, Nagarajan; Mambetsariev, Isa; Kindler, Hedy L; Wheeler, Deric L; Salgia, Ravi

Cooperation of neurotrophin receptor TrkB and Her2 in breast cancer cells facilitates brain metastases

神经营养因子受体TrkB和Her2在乳腺癌细胞中的协同作用促进脑转移

Choy, Cecilia; Ansari, Khairul I; Neman, Josh; Hsu, Sarah; Duenas, Matthew J; Li, Hubert; Vaidehi, Nagarajan; Jandial, Rahul

Human breast cancer metastases to the brain display GABAergic properties in the neural niche

人类乳腺癌脑转移灶在神经微环境中表现出GABA能特性。

Neman, Josh; Termini, John; Wilczynski, Sharon; Vaidehi, Nagarajan; Choy, Cecilia; Kowolik, Claudia M; Li, Hubert; Hambrecht, Amanda C; Roberts, Eugene; Jandial, Rahul

Critical analysis of the successes and failures of homology models of G protein-coupled receptors

对G蛋白偶联受体同源模型成功与失败的批判性分析

Bhattacharya, Supriyo; Lam, Alfonso Ramon; Li, Hubert; Balaraman, Gouthaman; Niesen, Michiel Jacobus Maria; Vaidehi, Nagarajan

Identification of anti-malarial compounds as novel antagonists to chemokine receptor CXCR4 in pancreatic cancer cells.

鉴定抗疟化合物为胰腺癌细胞中趋化因子受体 CXCR4 的新型拮抗剂

Kim Joseph, Yip M L Richard, Shen Xiaoming, Li Hubert, Hsin Li-Yu Charlie, Labarge Samuel, Heinrich Eileen L, Lee Wendy, Lu Jianming, Vaidehi Nagarajan

Ligand-stabilized conformational states of human beta(2) adrenergic receptor: insight into G-protein-coupled receptor activation

配体稳定的β2肾上腺素能受体构象状态:深入了解G蛋白偶联受体激活

Bhattacharya, Supriyo; Hall, Spencer E; Li, Hubert; Vaidehi, Nagarajan