日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Development and characterization of endolysosomal trafficking targeting chimera degraders of α(1A)-adrenergic receptor.

开发和表征靶向α(1A)-肾上腺素能受体嵌合降解剂的内溶酶体运输。

Chen Jiwei, Wang Shuo, Li Tong, Li Wenhua, Ke Xuechun, Ma Zhao, Du Lupei, Li Minyong

Erratum: Author correction to "Identification of anthelmintic parbendazole as a therapeutic molecule for HNSCC through connectivity map-based drug repositioning" [Acta Pharm Sin B 12 (2022) 2429-2442]

勘误:作者对“通过基于连接图的药物重定位鉴定抗蠕虫药帕苯达唑作为头颈部鳞状细胞癌的治疗分子”[Acta Pharm Sin B 12 (2022) 2429-2442]进行了更正。

Liang, Dong; Yu, Chen; Ma, Zhao; Yang, Xingye; Li, Zhenzhen; Dong, Xuhui; Qin, Xiaojun; Du, Lupei; Li, Minyong

Deuteration-Driven Photopharmacology: Deuterium-Labeled AzoCholine for Controlling Alpha 7 Nicotinic Acetylcholine Receptors

氘代驱动的光药理学:氘标记的偶氮胆碱用于控制α7尼古丁乙酰胆碱受体

Yang, Xingye; Zhou, Xin; Qin, Xiaojun; Liang, Dong; Dong, Xuhui; Ji, Huimin; Wen, Siman; Du, Lupei; Li, Minyong

Novel BRD4-p53 Inhibitor SDU-071 Suppresses Proliferation and Migration of MDA-MB-231 Triple-Negative Breast Cancer Cells.

新型 BRD4-p53 抑制剂 SDU-071 可抑制 MDA-MB-231 三阴性乳腺癌细胞的增殖和迁移

Wang Shumei, Lei Kang, Lai Hsien-Tsung, Liu Tingting, Du Lupei, Wu Shwu-Yuan, Ye Xiaohan, Chiang Cheng-Ming, Li Minyong

Engineered Bioluminescent Indicator Enables the Brain Imaging of Kinase Inhibitors

工程化生物发光指示剂可用于激酶抑制剂的脑成像

Ma, Zhao; Li, Minyong

Xuebijing Injection Attenuates Heat Stroke-Induced Brain Injury through Oxidative Stress Blockage and Parthanatos Modulation via PARP-1/AIF Signaling

血必净注射液通过阻断氧化应激和调节PARP-1/AIF信号转导减轻中暑引起的脑损伤

Lin Wang, Boxin Ye, Yongrui Liu, Jun Li, Chunhe Li, Minyong Wen, Hongbo Li

A pH-Driven Small-Molecule Nanotransformer Hijacks Lysosomes and Overcomes Autophagy-Induced Resistance in Cancer

一种pH驱动的小分子纳米转化器劫持溶酶体并克服癌症中自噬诱导的耐药性

Ma, Zhao; Lin, Kai; Tang, Menghuan; Ramachandran, Mythili; Qiu, Reng; Li, Jin; Solano, Lucas N; Huang, Yanyu; De Souza, Cristabelle; Abou-Adas, Sara; Xiang, Bai; Zhang, Lanwei; Li, Minyong; Li, Yuanpei

Fluorescent Ligand-Based Discovery of Small-Molecule Sulfonamide Agonists for GPR120

基于荧光配体的小分子磺酰胺类GPR120激动剂的发现

Ma, Siyue; Li, Zhenzhen; Yang, Yueli; Zhang, Ling; Li, Minyong; Du, Lupei

Author Correction: Pharmacophore hybridisation and nanoscale assembly to discover self-delivering lysosomotropic new-chemical entities for cancer therapy

作者更正:利用药效团杂交和纳米级组装技术发现用于癌症治疗的自递送溶酶体靶向新化学实体

Ma, Zhao; Li, Jin; Lin, Kai; Ramachandran, Mythili; Zhang, Dalin; Showalter, Megan; De Souza, Cristabelle; Lindstrom, Aaron; Solano, Lucas N; Jia, Bei; Urayama, Shiro; Duan, Yuyou; Fiehn, Oliver; Lin, Tzu-Yin; Li, Minyong; Li, Yuanpei

Visualization-Based Discovery of Vanin-1 Inhibitors for Colitis

基于可视化的Vanin-1抑制剂在结肠炎治疗中的发现

Wang, Guankai; Wang, Jingjing; Du, Lupei; Li, Minyong