日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of Niclosamide Analogs with Potent Mitochondrial Uncoupling Activity and Reduced Mitochondrial Inhibition-Associated Toxicity

发现具有强效线粒体解偶联活性和降低线粒体抑制相关毒性的尼克酰胺类似物

Jiang, Haowen; Macorano, Alessio; Xing, Enming; Jedoui, Mohamed; Mohammed, Shabber; Lee, Vanessa; Cheng, Jeffrey; McDonough, Lain; Cheng, Xiaolin; Ye, Jiangbin; Li, Pui Kai

Valine-Niclosamide for Treatment of Androgen Receptor Splice Variant-Positive Hepatocellular Carcinoma.

缬氨酸-尼克酰胺用于治疗雄激素受体剪接变异体阳性肝细胞癌

Hoelzen Emma J, Radomska Hanna S, Kulp Samuel K, Adeluola Adeoluwa A, Granchie Lauren A, Cheng Jeffrey, Dauki Anees M, Campbell Moray J, Mohammed Shabber, Xing Enming, Hai Min, Fukuda Mayu, Cheng Xiaolin, Phelps Mitch A, Li Pui-Kai, Coss Christopher C

Steroid Sulfatase Regulates Metabolic Reprogramming in Advanced Prostate Cancer.

类固醇硫酸酯酶调节晚期前列腺癌的代谢重编程

Sharifi Masuda, Armstrong Cameron M, Ning Shu, Leslie Amy R, Schaaf Zachary A, Maine James P, Lou Wei, Li Pui-Kai, Xu Hongyu, Liu Chengfei, Gao Allen C

Netupitant Exhibits Potent Activity on Mycobacterium tuberculosis Persisters

奈妥匹坦对结核分枝杆菌持续菌表现出强效活性

Eldesouky, Hassan E; Jones, Richard M; Mohammed, Shabber; Xing, Enming; Li, Pui-Kai; Sherman, David R

The pH gradient contributes to persistence in Mycobacterium tuberculosis

pH梯度有助于结核分枝杆菌的持续存在

Sherman, David; Eldesouky, Hassan; Adams, Kristin; Brache, Justin; Aguila, Laarni; Garcia, Mariana; Xing, Enming; Li, Pui-Kai

LX1 Dual Targets AR Variants and AKR1C3 in Advanced Prostate Cancer Therapy.

LX1 双靶点 AR 变异体和 AKR1C3 在晚期前列腺癌治疗中的应用

Ning Shu, Armstrong Cameron M, Xing Enming, Leslie Amy R, Gao Richard Y, Sharifi Masuda, Schaaf Zachary A, Lou Wei, Han Xiangrui, Xu Desiree H, Yang Rui, Cheng Jeffrey, Mohammed Shabber, Mitsiades Nicholas, Liu Chengfei, Lombard Alan P, Wu Chun-Yi, Cheng Xiaolin, Li Pui-Kai, Gao Allen C

Computational modeling studies reveal the origin of the binding preference of 3-(3,4-di hydroisoquinolin-2(1H)-ylsulfonyl)benzoic acids for AKR1C3 over its isoforms

计算模型研究揭示了 3-(3,4-二氢异喹啉-2(1H)-基磺酰基)苯甲酸对 AKR1C3 的结合偏好性高于其同工酶的起源

Kong, Xiaotian; Xing, Enming; Wu, Sijin; Zhuang, Tony; Li, Pui-Kai; Li, Chunhua; Cheng, Xiaolin

Correction: Niclosamide and its analogs are potent inhibitors of Wnt/β-catenin, mTOR and STAT3 signaling in ovarian cancer

更正:尼克酰胺及其类似物是卵巢癌中Wnt/β-catenin、mTOR和STAT3信号通路的强效抑制剂。

Arend, Rebecca C; Londoño-Joshi, Angelina I; Gangrade, Abhishek; Katre, Ashwini A; Kurpad, Chandrika; Li, Yonghe; Samant, Rajeev S; Li, Pui-Kai; Landen, Charles N; Yang, Eddy S; Hidalgo, Bertha; Alvarez, Ronald D; Straughn, John Michael; Forero, Andres; Buchsbaum, Donald J

Protective effect of suppressing STAT3 activity in LPS-induced acute lung injury

抑制STAT3活性对LPS诱导的急性肺损伤的保护作用

Zhao, Jiping; Yu, Hao; Liu, Yudong; Gibson, Sara A; Yan, Zhaoqi; Xu, Xin; Gaggar, Amit; Li, Pui-Kai; Li, Chenglong; Wei, Shi; Benveniste, Etty N; Qin, Hongwei

Niclosamide and its analogs are potent inhibitors of Wnt/β-catenin, mTOR and STAT3 signaling in ovarian cancer.

尼克酰胺及其类似物是卵巢癌中 Wnt/β-catenin、mTOR 和 STAT3 信号传导的强效抑制剂

Arend Rebecca C, Londoño-Joshi Angelina I, Gangrade Abhishek, Katre Ashwini A, Kurpad Chandrika, Li Yonghe, Samant Rajeev S, Li Pui-Kai, Landen Charles N, Yang Eddy S, Hidalgo Bertha, Alvarez Ronald D, Straughn John Michael, Forero Andres, Buchsbaum Donald J