Discovery of peptidomimetic inhibitors of CREB/CBP by targeting hydrophobic grooves on the surface of the CBP KIX domain
通过靶向CBP KIX结构域表面的疏水沟槽,发现CREB/CBP的肽模拟抑制剂。
期刊:Acta Pharmaceutica Sinica B
影响因子:14.6
doi:10.1016/j.apsb.2025.08.023
Huang, Bo; Gregory-Lott, Emily; Li, Bingbing X; Tran, Timothy H; Li, Sihao; Xue, Menglin; Wang, Shaohui; Asokan, Anabanadam; Shen, Ning; Sun, Xingming; Cao, Chuanhai; Xiao, Xiangshu; Daughdrill, Gary; Cai, Jianfeng