日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design and characterization of a potent and selective dual ATP- and substrate-competitive subnanomolar bidentate c-Jun N-terminal kinase (JNK) inhibitor

设计和表征一种强效且选择性双重 ATP 和底物竞争性亚纳摩尔双齿 c-Jun N 端激酶 (JNK) 抑制剂

John L Stebbins, Surya K De, Petra Pavlickova, Vida Chen, Thomas Machleidt, Li-Hsing Chen, Christian Kuntzen, Shinichi Kitada, Michael Karin, Maurizio Pellecchia

Targeting metalloproteins by fragment-based lead discovery

通过基于片段的先导化合物发现靶向金属蛋白

Sherida Johnson, Elisa Barile, Biancamaria Farina, Angela Purves, Jun Wei, Li-Hsing Chen, Sergey Shiryaev, Ziming Zhang, Irina Rodionova, Arpita Agrawal, Seth M Cohen, Andrei Osterman, Alex Strongin, Maurizio Pellecchia

Design, synthesis, and structure-activity relationship of substrate competitive, selective, and in vivo active triazole and thiadiazole inhibitors of the c-Jun N-terminal kinase

底物竞争性、选择性和体内活性的 c-Jun N 端激酶三唑和噻二唑抑制剂的设计、合成和构效关系

Surya K De, John L Stebbins, Li-Hsing Chen, Megan Riel-Mehan, Thomas Machleidt, Russell Dahl, Hongbin Yuan, Aras Emdadi, Elisa Barile, Vida Chen, Ria Murphy, Maurizio Pellecchia